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Schema
>
LiteratureReference
>
Entries
Complementary activity of tyrosine kinase inhibitors against secondary kit mutations in imatinib-resistant gastrointestinal stromal tumours
Show undefined attributes
author
[Person:9669090] Serrano, C
[Person:9669080] Mariño-Enríquez, A
[Person:9669085] Tao, DL
[Person:9669097] Ketzer, J
[Person:9669082] Eilers, G
[Person:9669092] Zhu, M
[Person:9669091] Yu, C
[Person:9669089] Mannan, AM
[Person:9669086] Rubin, BP
[Person:9669081] Demetri, GD
[Person:9669095] Raut, CP
[Person:9669093] Presnell, A
[Person:9669079] McKinley, A
[Person:9669096] Heinrich, MC
[Person:9669078] Czaplinski, JT
[Person:9669084] Sicinska, E
[Person:9669098] Bauer, S
[Person:9669088] George, S
[Person:9669087] Fletcher, JA
created
[InstanceEdit:9669083] Rothfels, Karen, 2019-12-02
dbId
9669094
displayName
Complementary activity of tyrosine kinase inhibitors against secondary kit mutations in imatinib-resistant gastrointestinal stromal tumours
journal
Br. J. Cancer
pages
612-620
pubMedIdentifier
30792533
schemaClass
LiteratureReference
title
Complementary activity of tyrosine kinase inhibitors against secondary kit mutations in imatinib-resistant gastrointestinal stromal tumours
url
http://www.ncbi.nlm.nih.gov/pubmed/30792533
volume
120
year
2019
Referrals
(literatureReference)
[Pathway:R-HSA-9669933] Signaling by kinase domain mutants of KIT
[Reaction:R-HSA-9670433] KIT mutants:PI3K catalyze synthesis of PIP3
[EntityWithAccessionedSequence:R-HSA-9670336] KIT V560_L576del [plasma membrane]
[Pathway:R-HSA-9669937] Drug resistance of KIT mutants
[Pathway:R-HSA-9669917] Imatinib-resistant KIT mutants
[FailedReaction:R-HSA-9669859] Imatinib-resistant KIT mutants do not bind imatinib
[FailedReaction:R-HSA-9669878] Sunitinib-resistant KIT mutants do not bind sunitinib
[Pathway:R-HSA-9669929] Regorafenib-resistant KIT mutants
[FailedReaction:R-HSA-9669870] Regorafenib-resistant KIT mutants do not bind regorafenib
[Pathway:R-HSA-9669914] Dasatinib-resistant KIT mutants
[FailedReaction:R-HSA-9669855] Dasatinib-resistant KIT mutants do not bind dasatinib
[Pathway:R-HSA-9669924] Masitinib-resistant KIT mutants
[FailedReaction:R-HSA-9669863] Masitinib-resistant KIT mutants do not bind masitinib
[Pathway:R-HSA-9669926] Nilotinib-resistant KIT mutants
[FailedReaction:R-HSA-9669868] Nilotinib-resistant KIT mutants do not bind nilotinib
[DefinedSet:R-HSA-9669772] nilotinib resistant KIT mutants [plasma membrane]
[Pathway:R-HSA-9669936] Sorafenib-resistant KIT mutants
[FailedReaction:R-HSA-9669874] Sorafenib-resistant KIT mutants do not bind sorafenib
[Pathway:R-HSA-9669921] KIT mutants bind TKIs
[Reaction:R-HSA-9669900] KIT mutants bind type II TKIs
[DefinedSet:R-HSA-9669750] imatinib sensitive KIT mutants [plasma membrane]
[Reaction:R-HSA-9669898] KIT mutants bind type I TKIs
[DefinedSet:R-HSA-9669742] dovitinib sensitive KIT mutants [plasma membrane]
[EntityWithAccessionedSequence:R-HSA-9670343] KIT W557_K558del [plasma membrane]
[RegulationReference:9669883] Negative regulation by 'KIT:sSCF dimer:KIT:type I KIT binding TKIs: [plasma membrane]' Complementary activity of tyrosine kinase inhibitors against secondary kit mutations in imatinib-resistant gastrointestinal stromal tumours
(author)
[Person:9669096] Heinrich, MC
[Person:9669097] Ketzer, J
[Person:9669098] Bauer, S
[Person:9669092] Zhu, M
[Person:9669093] Presnell, A
[Person:9669095] Raut, CP
[Person:9669088] George, S
[Person:9669089] Mannan, AM
[Person:9669090] Serrano, C
[Person:9669091] Yu, C
[Person:9669084] Sicinska, E
[Person:9669085] Tao, DL
[Person:9669086] Rubin, BP
[Person:9669087] Fletcher, JA
[Person:9669080] Mariño-Enríquez, A
[Person:9669081] Demetri, GD
[Person:9669082] Eilers, G
[Person:9669078] Czaplinski, JT
[Person:9669079] McKinley, A
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