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Search ...
Go!
Schema
>
ChemicalDrug
>
Entries
dovitinib [cytosol]
Show undefined attributes
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compartment
[Compartment:70101] cytosol
created
[InstanceEdit:1839034] Rothfels, K, 2011-10-27
crossReference
[DatabaseIdentifier:9628078] PubChem Compound:9886808
dbId
1839035
disease
[Disease:1500689] cancer
displayName
dovitinib [cytosol]
inDisease
true
literatureReference
[LiteratureReference:2023313] In vivo target modulation and biological activity of CHIR-258, a multitargeted growth factor receptor kinase inhibitor, in colon cancer models
[LiteratureReference:2023310] A phase I pharmacokinetic and pharmacodynamic study of TKI258, an oral, multitargeted receptor tyrosine kinase inhibitor in patients with advanced solid tumors
memberOf
[DefinedSet:R-ALL-2023441] Tyrosine kinase inhibitors of overexpressed FGFR1 [cytosol]
[DefinedSet:R-ALL-2045079] Tyrosine kinase inhibitors of FGFR1 fusion mutants [cytosol]
[DefinedSet:R-ALL-9669710] type I KIT binding TKIs [cytosol]
[DefinedSet:R-ALL-2077416] Tyrosine kinase inhibitors of FGFR3 mutants [cytosol]
modified
[InstanceEdit:9669664] Rothfels, Karen, 2019-12-03
name
dovitinib
TKI258
referenceEntity
[ReferenceTherapeutic:9603941] dovitinib [Guide to Pharmacology:5962]
schemaClass
ChemicalDrug
stId
R-ALL-1839035
summation
[Summation:2023211] A Novartis tyrosine kinase inhibitor with activity against m...
Referrals
(hasMember)
[DefinedSet:R-ALL-2077416] Tyrosine kinase inhibitors of FGFR3 mutants [cytosol]
[DefinedSet:R-ALL-2023441] Tyrosine kinase inhibitors of overexpressed FGFR1 [cytosol]
[DefinedSet:R-ALL-2045079] Tyrosine kinase inhibitors of FGFR1 fusion mutants [cytosol]
[DefinedSet:R-ALL-9669710] type I KIT binding TKIs [cytosol]
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