The following FLT3 mutants are resistant to inhibition by semaxanib: FLT3 D835N (partial: Bagrintseva et al, 2005) FLT3 D835Y (partial: Bagrintseva et al, 2005)
Ellwart, JW, Reindl, C, Spiekermann, K, Geisenhof, S, Kern, R, Bagrintseva, K, Hiddemann, W, Eichenlaub, S
Loss of function of semaxanib-resistant FLT3 mutants [plasma membrane]
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