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CYSLTR1 [plasma membrane]
Stable Identifier
R-HSA-416418
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
plasma membrane
Synonyms
Cysteinyl leukotriene receptor 1, CLTR1_HUMAN
Locations in the PathwayBrowser
Expand all
Disease (Homo sapiens)
Infectious disease (Homo sapiens)
Parasitic Infection Pathways (Homo sapiens)
Leishmania infection (Homo sapiens)
Leishmania parasite growth and survival (Homo sapiens)
Anti-inflammatory response favouring Leishmania parasite infection (Homo sapiens)
LTC4-CYSLTR mediated IL4 production (Homo sapiens)
LTC4 binds CyslTR1,2 (Homo sapiens)
CYSLTR1,CYSLTR2 [plasma membrane] (Homo sapiens)
CYSLTR1 [plasma membrane] (Homo sapiens)
LTC4:CyslTR1,2 [plasma membrane] (Homo sapiens)
CYSLTR1,CYSLTR2 [plasma membrane] (Homo sapiens)
CYSLTR1 [plasma membrane] (Homo sapiens)
Viral Infection Pathways (Homo sapiens)
SARS-CoV Infections (Homo sapiens)
Potential therapeutics for SARS (Homo sapiens)
CYSLTR1 binds CYSLTR1 antagonists (Homo sapiens)
CYSLTR1 [plasma membrane] (Homo sapiens)
CYSLTR1:CYSLTR1 antagonists [plasma membrane] (Homo sapiens)
CYSLTR1 [plasma membrane] (Homo sapiens)
Signal Transduction (Homo sapiens)
Signaling by GPCR (Homo sapiens)
GPCR downstream signalling (Homo sapiens)
G alpha (q) signalling events (Homo sapiens)
Liganded Gq-activating GPCRs bind inactive heterotrimeric Gq (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
CYSLTR1:LTC4,LTD4,LTE4 [plasma membrane] (Homo sapiens)
CYSLTR1 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
CYSLTR1:LTC4,LTD4,LTE4 [plasma membrane] (Homo sapiens)
CYSLTR1 [plasma membrane] (Homo sapiens)
Liganded Gq/11-activating GPCRs act as GEFs for Gq/11 (Homo sapiens)
LTC4:CyslTR1,2 [plasma membrane] (Homo sapiens)
CYSLTR1,CYSLTR2 [plasma membrane] (Homo sapiens)
CYSLTR1 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
CYSLTR1:LTC4,LTD4,LTE4 [plasma membrane] (Homo sapiens)
CYSLTR1 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
CYSLTR1:LTC4,LTD4,LTE4 [plasma membrane] (Homo sapiens)
CYSLTR1 [plasma membrane] (Homo sapiens)
The Ligand:GPCR:Gq complex dissociates (Homo sapiens)
GPCRs that activate Gq/11 [plasma membrane] (Homo sapiens)
CYSLTR1 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
CYSLTR1:LTC4,LTD4,LTE4 [plasma membrane] (Homo sapiens)
CYSLTR1 [plasma membrane] (Homo sapiens)
GPCR ligand binding (Homo sapiens)
Class A/1 (Rhodopsin-like receptors) (Homo sapiens)
Eicosanoid ligand-binding receptors (Homo sapiens)
Leukotriene receptors (Homo sapiens)
CYSLTR1 binds CYSLTR1 antagonists (Homo sapiens)
CYSLTR1 [plasma membrane] (Homo sapiens)
CYSLTR1:CYSLTR1 antagonists [plasma membrane] (Homo sapiens)
CYSLTR1 [plasma membrane] (Homo sapiens)
CYSLTR1 binds LTC4,LTD4,LTE4 (Homo sapiens)
CYSLTR1 [plasma membrane] (Homo sapiens)
CYSLTR1:CYSLTR1 antagonists [plasma membrane] (Homo sapiens)
CYSLTR1 [plasma membrane] (Homo sapiens)
CYSLTR1:LTC4,LTD4,LTE4 [plasma membrane] (Homo sapiens)
CYSLTR1 [plasma membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:Q9Y271 CYSLTR1
Gene Names
CYSLTR1, CYSLT1
Chain
chain:1-337
Reference Genes
BioGPS Gene:10800 CYSLTR1
COSMIC (genes):CYSLTR1 CYSLTR1
CTD Gene:10800 CYSLTR1
dbSNP Gene:10800 CYSLTR1
ENSEMBL:ENSG00000173198 CYSLTR1
HGNC:17451 CYSLTR1
KEGG:hsa:10800 CYSLTR1
Monarch:10800 CYSLTR1
NCBI Gene:10800 CYSLTR1
OMIM:300201 CYSLTR1
UCSC:Q9Y271 CYSLTR1
Reference Transcript
RefSeq:NM_001282187.1 CYSLTR1
RefSeq:NM_001282188.1 CYSLTR1
RefSeq:NM_001282186.1 CYSLTR1
RefSeq:NM_006639.3 CYSLTR1
Other Identifiers
10800
11735157_at
11759152_at
17112349
216288_PM_at
216288_at
230866_PM_at
230866_at
231747_PM_at
231747_at
4013461
4013462
4013463
4013464
4013465
4013466
4013467
4013468
4013471
4013472
4013474
81554_at
8173745
A_23_P22660
A_24_P915225
GE58410
GO:0001631
GO:0002376
GO:0002437
GO:0003013
GO:0004930
GO:0004974
GO:0005886
GO:0006816
GO:0006935
GO:0006952
GO:0006954
GO:0007166
GO:0007186
GO:0007204
GO:0007218
GO:0007585
GO:0008528
GO:0016020
GO:0045766
GO:0045907
GO:0051649
GO:0060089
GO:0060252
GO:0061737
GO:0071456
HMNXSV003042093
Hs.121139.0.A1_3p_at
Hs.124401.0.S1_3p_at
Hs.301150.0.S1_3p_at
ILMN_1733276
PH_hs_0022985
TC0X001177.hg
Participates
as an input of
CYSLTR1 binds CYSLTR1 antagonists (Homo sapiens)
CYSLTR1 binds LTC4,LTD4,LTE4 (Homo sapiens)
as a component of
CYSLTR1:CYSLTR1 antagonists [plasma membrane] (Homo sapiens)
CYSLTR1:LTC4,LTD4,LTE4 [plasma membrane] (Homo sapiens)
as a member of
CYSLTR1,CYSLTR2 [plasma membrane] (Homo sapiens)
GPCRs that activate Gq/11 [plasma membrane] (Homo sapiens)
Inferred To
AstA-R2 [plasma membrane]
(Drosophila melanogaster)
CYSLTR1 [plasma membrane]
(Bos taurus)
CYSLTR1 [plasma membrane]
(Canis familiaris)
CYSLTR1 [plasma membrane]
(Gallus gallus)
CYSLTR1 [plasma membrane]
(Sus scrofa)
cysltr1 [plasma membrane]
(Danio rerio)
Cysltr1 [plasma membrane]
(Mus musculus)
Cysltr1 [plasma membrane]
(Rattus norvegicus)
Homologues of CYSLTR1 [plasma membrane]
(Drosophila melanogaster)
npr-14 [plasma membrane]
(Caenorhabditis elegans)
CG 13579 [plasma membrane]
(Drosophila melanogaster)
Cross References
RefSeq
NP_006630.1
,
NP_001269115.1
,
NP_001269117.1
,
NP_001269116.1
Guide to Pharmacology - Targets
269
ENSEMBL
ENSG00000173198
,
ENST00000373304
,
ENSP00000362401
,
ENSP00000478492
,
ENST00000614798
OpenTargets
ENSG00000173198
ZINC - FDA approved
CLTR1_HUMAN
ZINC - Substances
CLTR1_HUMAN
ZINC - Biogenic
CLTR1_HUMAN
ZINC target
Q9Y271
PRO
Q9Y271
GlyGen
Q9Y271
PDB
6RZ4
,
6RZ5
ZINC - Investigational
CLTR1_HUMAN
ZINC - Metabolites
CLTR1_HUMAN
GeneCards
CYSLTR1
HPA
ENSG00000173198-CYSLTR1
Pharos - Targets
Q9Y271
ZINC - Predictions - Purchasable
CLTR1_HUMAN
HMDB Protein
HMDBP02258
Interactors (1)
Accession
#Entities
Entities
Confidence Score
Evidence (IntAct)
UniProt:Q9NS75 CYSLTR2
1
CYSLTR2 [plasma membrane]
(R-HSA-416399)
0.471
2
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