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Reaction
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Entries
Dimerization of FGFR1 point mutants with enhanced kinase activity
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authored
[InstanceEdit:2105031] Rothfels, K, 2012-02-09
category
transition
compartment
[Compartment:876] plasma membrane
created
[InstanceEdit:2023457] Rothfels, K, 2011-12-07
dbId
2023456
disease
[Disease:1500689] cancer
[Disease:2011833] glioblastoma
displayName
Dimerization of FGFR1 point mutants with enhanced kinase activity
edited
[InstanceEdit:2252592] Rothfels, K, 2012-05-16
entityFunctionalStatus
[EntityFunctionalStatus:5654486] gain_of_function of FGFR1 mutants with enhanced kinase activity [plasma membrane]
eventOf
[Pathway:R-HSA-1839122] Signaling by activated point mutants of FGFR1 - Homo sapiens
followingEvent
[Reaction:R-HSA-2023460] Autocatalytic phosphorylation of FGFR1 mutants with enhanced kinase activity - Homo sapiens
input
2 ×
[CandidateSet:R-HSA-2012030] FGFR1 mutants with enhanced kinase activity [plasma membrane]
isChimeric
false
isInDisease
true
isInferred
false
literatureReference
[LiteratureReference:1614276] The precise sequence of FGF receptor autophosphorylation is kinetically driven and is disrupted by oncogenic mutations
[LiteratureReference:1614269] Sequence survey of receptor tyrosine kinases reveals mutations in glioblastomas
[LiteratureReference:1295608] Transformation and Stat activation by derivatives of FGFR1, FGFR3, and FGFR4
[LiteratureReference:2012013] Induction of chondrogenesis in neural crest cells by mutant fibroblast growth factor receptors
[LiteratureReference:1614246] Comprehensive genomic characterization defines human glioblastoma genes and core pathways
[LiteratureReference:2054036] Effect of transmembrane and kinase domain mutations on fibroblast growth factor receptor 3 chimera signaling in PC12 cells. A model for the control of receptor tyrosine kinase activation
modified
[InstanceEdit:9830342] Matthews, Lisa, 2023-03-08
name
Dimerization of FGFR1 point mutants with enhanced kinase activity
output
[CandidateSet:R-HSA-2023433] FGFR1 mutant dimers with enhanced kinase activity [plasma membrane]
releaseDate
2012-06-12
reviewStatus
[ReviewStatus:9821382] five stars
reviewed
[InstanceEdit:2248845] Ezzat, S, 2012-05-15
schemaClass
Reaction
species
[Species:48887] Homo sapiens
stId
R-HSA-2023456
summation
[Summation:2054043] Large scale genomic characterization of glioblastoma tumors ...
Referrals
(hasEvent)
[Pathway:R-HSA-1839122] Signaling by activated point mutants of FGFR1
(precedingEvent)
[Reaction:R-HSA-2023460] Autocatalytic phosphorylation of FGFR1 mutants with enhanced kinase activity
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