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ADRA1D [plasma membrane]
Stable Identifier
R-HSA-390680
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
plasma membrane
Synonyms
Alpha-1D adrenoceptor, RecName: Full=Alpha-1D adrenergic receptor; AltName: Full=Alpha 1D-adrenoreceptor; AltName: Full=Alpha 1D-adrenoceptor; AltName: Full=Alpha-1A adrenergic receptor; AltName: Full=Alpha-adrenergic receptor 1a;
GN Name=ADRA1D; Synonyms=ADRA1A;
OS Homo sapiens, ADA1D_HUMAN
Locations in the PathwayBrowser
Expand all
Signal Transduction (Homo sapiens)
Signaling by GPCR (Homo sapiens)
GPCR downstream signalling (Homo sapiens)
G alpha (12/13) signalling events (Homo sapiens)
Liganded G12/13-activating GPCR acts as a GEF for G12/13 (Homo sapiens)
Ligand:GPCR complexes that activate G12/13:Heterotrimeric G-protein G12/13 (active). [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate G12/13 [plasma membrane] (Homo sapiens)
ADRA1A,B,D:ADR,NAd [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1D [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate G12/13:Heterotrimeric G-protein G12/13 (inactive). [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate G12/13 [plasma membrane] (Homo sapiens)
ADRA1A,B,D:ADR,NAd [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1D [plasma membrane] (Homo sapiens)
Liganded G12/13-activating GPCRs bind inactive heterotrimeric G-protein G12/13 (Homo sapiens)
Ligand:GPCR complexes that activate G12/13 [plasma membrane] (Homo sapiens)
ADRA1A,B,D:ADR,NAd [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1D [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate G12/13:Heterotrimeric G-protein G12/13 (inactive). [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate G12/13 [plasma membrane] (Homo sapiens)
ADRA1A,B,D:ADR,NAd [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1D [plasma membrane] (Homo sapiens)
The Ligand:GPCR:G12/13 complex dissociates (Homo sapiens)
GPCRs that activate G12/13 [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1D [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate G12/13:Heterotrimeric G-protein G12/13 (active). [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate G12/13 [plasma membrane] (Homo sapiens)
ADRA1A,B,D:ADR,NAd [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1D [plasma membrane] (Homo sapiens)
G alpha (q) signalling events (Homo sapiens)
Liganded Gq-activating GPCRs bind inactive heterotrimeric Gq (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
ADRA1A,B,D:ADR,NAd [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1D [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
ADRA1A,B,D:ADR,NAd [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1D [plasma membrane] (Homo sapiens)
Liganded Gq/11-activating GPCRs act as GEFs for Gq/11 (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
ADRA1A,B,D:ADR,NAd [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1D [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
ADRA1A,B,D:ADR,NAd [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1D [plasma membrane] (Homo sapiens)
The Ligand:GPCR:Gq complex dissociates (Homo sapiens)
GPCRs that activate Gq/11 [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1D [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
ADRA1A,B,D:ADR,NAd [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1D [plasma membrane] (Homo sapiens)
GPCR ligand binding (Homo sapiens)
Class A/1 (Rhodopsin-like receptors) (Homo sapiens)
Amine ligand-binding receptors (Homo sapiens)
Adrenoceptors (Homo sapiens)
ADRA1A,B,D bind ADR,NAd (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1D [plasma membrane] (Homo sapiens)
ADRA1A,B,D:ADR,NAd [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1D [plasma membrane] (Homo sapiens)
α1-agonists:ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1D [plasma membrane] (Homo sapiens)
α1-antagonists:ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1D [plasma membrane] (Homo sapiens)
α1-agonists bind ADRA1A,B,D (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1D [plasma membrane] (Homo sapiens)
α1-agonists:ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1D [plasma membrane] (Homo sapiens)
α1-antagonists bind ADRA1A,B,D (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1D [plasma membrane] (Homo sapiens)
α1-antagonists:ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1D [plasma membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:P25100 ADRA1D
Gene Names
ADRA1D, ADRA1A
Chain
chain:1-572
Reference Genes
BioGPS Gene:146 ADRA1D
COSMIC (genes):ADRA1D ADRA1D
CTD Gene:146 ADRA1D
dbSNP Gene:146 ADRA1D
ENSEMBL:ENSG00000171873 ADRA1D
ENSEMBL_homo_sapiens_GENE:ENSG00000171873.8 ADRA1D
HGNC:280 ADRA1D
KEGG Gene (Homo sapiens):146 ADRA1D
Monarch:146 ADRA1D
NCBI Gene:146 ADRA1D
OMIM:104219 ADRA1D
UCSC:P25100 ADRA1D
Reference Transcript
RefSeq:NM_000678.3 ADRA1D
Other Identifiers
11740618_at
11740619_at
146
16916877
210960_PM_at
210960_at
210961_PM_s_at
210961_s_at
36728_at
36729_g_at
3895892
3895893
3895894
3895902
3895903
3895904
3895905
3895906
8064779
90822_at
A_23_P131924
A_33_P3243023
GE62553
GO:0003013
GO:0004930
GO:0004935
GO:0004937
GO:0005515
GO:0005886
GO:0007165
GO:0007186
GO:0007188
GO:0007200
GO:0007204
GO:0007267
GO:0008284
GO:0016020
GO:0023052
GO:0042802
GO:0045907
GO:0060089
GO:0071875
GO:0071880
GO:0150099
HMNXSV003030075
ILMN_1716421
M76446_at
PH_hs_0000065
TC20000584.hg
g177806_3p_at
Participates
as a member of
ADRA1A,B,D [plasma membrane] (Homo sapiens)
Inferred To
ser-5 [plasma membrane]
(Caenorhabditis elegans)
Adra1d [plasma membrane]
(Mus musculus)
Adra1d [plasma membrane]
(Rattus norvegicus)
Homologues of ADRA1D [plasma membrane]
(Sus scrofa)
ADRA1D [plasma membrane]
(Bos taurus)
ADRA1D [plasma membrane]
(Canis familiaris)
ADRA1D [plasma membrane]
(Gallus gallus)
ADRA1D [plasma membrane]
(Sus scrofa)
DopEcR [plasma membrane]
(Drosophila melanogaster)
Cross References
RefSeq
NP_000669.1
ZINC - World Drugs
ADA1D_HUMAN
Guide to Pharmacology - Targets
24
OpenTargets
ENSG00000171873
ZINC - FDA approved
ADA1D_HUMAN
ZINC - Substances
ADA1D_HUMAN
ZINC target
P25100
ZINC - Biogenic
ADA1D_HUMAN
PRO
P25100
ZINC - Investigational
ADA1D_HUMAN
ZINC - Metabolites
ADA1D_HUMAN
HPA
ENSG00000171873-ADRA1D
GeneCards
P25100
Ensembl
ENSP00000368766
,
ENST00000379453
,
ENSG00000171873
Pharos - Targets
P25100
ZINC - Predictions - Purchasable
ADA1D_HUMAN
HMDB Protein
HMDBP07435
Interactors (3)
Accession
#Entities
Entities
Confidence Score
Evidence (IntAct)
UniProt:P46939 UTRN
1
UTRN [cytosol]
(R-HSA-5216039)
0.773
14
UniProt:Q14160 SCRIB
1
SCRIB [cytosol]
(R-HSA-4608858)
0.76
19
UniProt:P11532 DMD
1
DMD [cytosol]
(R-HSA-390567)
0.527
8
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