Atorvastatin (ATV) is hydroxylated to hydroxy-metabolites, p...

created [InstanceEdit:9756787] Jassal, Bijay, 2021-10-18
dbId 9756792
displayName Atorvastatin (ATV) is hydroxylated to hydroxy-metabolites, p...
modified [InstanceEdit:9757281] Jassal, Bijay, 2021-10-28
schemaClass Summation
text Atorvastatin (ATV) is hydroxylated to hydroxy-metabolites, predominantly by cytochrome P450 3A4 (CYP3A4) (Fujino et al. 2004, Park et al. 2008). Here, ATV hydroxylation to 4-hydroxyatorvastatin (4-OH-ATV, aka para-hydroxyatorvastatin) is described.
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