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SGX-523 [cytosol]
Stable Identifier
R-ALL-9735966
Type
ChemicalDrug
Compartment
cytosol
Locations in the PathwayBrowser
for Species:
Homo sapiens
Bos taurus
Canis familiaris
Danio rerio
Gallus gallus
Mus musculus
Rattus norvegicus
Sus scrofa
Xenopus tropicalis
Expand all
Signal Transduction (Bos taurus)
Signaling by Receptor Tyrosine Kinases (Bos taurus)
Signaling by MET (Bos taurus)
MET Receptor Activation (Bos taurus)
MET dimers autophosphorylate (Bos taurus)
HGF:MET dimer:TKIs [plasma membrane] (Bos taurus)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
Negative regulation of MET activity (Bos taurus)
Drug-mediated inhibition of MET activation (Bos taurus)
Anti-MET small tyrosine kinase inhibitors bind MET (Bos taurus)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
HGF:MET dimer:TKIs [plasma membrane] (Bos taurus)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
Signal Transduction (Canis familiaris)
Signaling by Receptor Tyrosine Kinases (Canis familiaris)
Signaling by MET (Canis familiaris)
MET Receptor Activation (Canis familiaris)
MET dimers autophosphorylate (Canis familiaris)
HGF:MET dimer:TKIs [plasma membrane] (Canis familiaris)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
Negative regulation of MET activity (Canis familiaris)
Drug-mediated inhibition of MET activation (Canis familiaris)
Anti-MET small tyrosine kinase inhibitors bind MET (Canis familiaris)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
HGF:MET dimer:TKIs [plasma membrane] (Canis familiaris)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
Signal Transduction (Danio rerio)
Signaling by Receptor Tyrosine Kinases (Danio rerio)
Signaling by MET (Danio rerio)
MET Receptor Activation (Danio rerio)
MET dimers autophosphorylate (Danio rerio)
HGF:MET dimer:TKIs [plasma membrane] (Danio rerio)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
Negative regulation of MET activity (Danio rerio)
Drug-mediated inhibition of MET activation (Danio rerio)
Anti-MET small tyrosine kinase inhibitors bind MET (Danio rerio)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
HGF:MET dimer:TKIs [plasma membrane] (Danio rerio)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
Signal Transduction (Gallus gallus)
Signaling by Receptor Tyrosine Kinases (Gallus gallus)
Signaling by MET (Gallus gallus)
MET Receptor Activation (Gallus gallus)
MET dimers autophosphorylate (Gallus gallus)
HGF:MET dimer:TKIs [plasma membrane] (Gallus gallus)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
Negative regulation of MET activity (Gallus gallus)
Drug-mediated inhibition of MET activation (Gallus gallus)
Anti-MET small tyrosine kinase inhibitors bind MET (Gallus gallus)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
HGF:MET dimer:TKIs [plasma membrane] (Gallus gallus)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
Signal Transduction (Homo sapiens)
Signaling by Receptor Tyrosine Kinases (Homo sapiens)
Signaling by MET (Homo sapiens)
MET Receptor Activation (Homo sapiens)
MET dimers autophosphorylate (Homo sapiens)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
HGF:MET dimer:TKIs [plasma membrane] (Homo sapiens)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
Negative regulation of MET activity (Homo sapiens)
Drug-mediated inhibition of MET activation (Homo sapiens)
Anti-MET small tyrosine kinase inhibitors bind MET (Homo sapiens)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
HGF:MET dimer:TKIs [plasma membrane] (Homo sapiens)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
Signal Transduction (Mus musculus)
Signaling by Receptor Tyrosine Kinases (Mus musculus)
Signaling by MET (Mus musculus)
MET Receptor Activation (Mus musculus)
MET dimers autophosphorylate (Mus musculus)
HGF:MET dimer:TKIs [plasma membrane] (Mus musculus)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
Negative regulation of MET activity (Mus musculus)
Drug-mediated inhibition of MET activation (Mus musculus)
Anti-MET small tyrosine kinase inhibitors bind MET (Mus musculus)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
HGF:MET dimer:TKIs [plasma membrane] (Mus musculus)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
Signal Transduction (Rattus norvegicus)
Signaling by Receptor Tyrosine Kinases (Rattus norvegicus)
Signaling by MET (Rattus norvegicus)
MET Receptor Activation (Rattus norvegicus)
MET dimers autophosphorylate (Rattus norvegicus)
HGF:MET dimer:TKIs [plasma membrane] (Rattus norvegicus)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
Negative regulation of MET activity (Rattus norvegicus)
Drug-mediated inhibition of MET activation (Rattus norvegicus)
Anti-MET small tyrosine kinase inhibitors bind MET (Rattus norvegicus)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
HGF:MET dimer:TKIs [plasma membrane] (Rattus norvegicus)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
Signal Transduction (Sus scrofa)
Signaling by Receptor Tyrosine Kinases (Sus scrofa)
Signaling by MET (Sus scrofa)
MET Receptor Activation (Sus scrofa)
MET dimers autophosphorylate (Sus scrofa)
HGF:MET dimer:TKIs [plasma membrane] (Sus scrofa)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
Negative regulation of MET activity (Sus scrofa)
Drug-mediated inhibition of MET activation (Sus scrofa)
Anti-MET small tyrosine kinase inhibitors bind MET (Sus scrofa)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
HGF:MET dimer:TKIs [plasma membrane] (Sus scrofa)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
Signal Transduction (Xenopus tropicalis)
Signaling by Receptor Tyrosine Kinases (Xenopus tropicalis)
Signaling by MET (Xenopus tropicalis)
MET Receptor Activation (Xenopus tropicalis)
MET dimers autophosphorylate (Xenopus tropicalis)
HGF:MET dimer:TKIs [plasma membrane] (Xenopus tropicalis)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
Negative regulation of MET activity (Xenopus tropicalis)
Drug-mediated inhibition of MET activation (Xenopus tropicalis)
Anti-MET small tyrosine kinase inhibitors bind MET (Xenopus tropicalis)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
HGF:MET dimer:TKIs [plasma membrane] (Xenopus tropicalis)
Anti-MET TKIs [cytosol]
SGX-523 [cytosol]
External Reference Information
External Reference
SGX-523 [Guide to Pharmacology:5709]
Participates
as a member of
Anti-MET TKIs [cytosol]
Disease
Name
Identifier
Synonyms
cancer
DOID:162
malignant tumor, malignant neoplasm, primary cancer
Cross References
Mondo
0004992
ChEBI
90624
PharmacoDB
PDBC01878
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