The following FLT3 mutants are resistant to tamatinib-mediated inhibition:FLT3 Y591_V592insVDFREYEYDH (Nguyen et al, 2017) FLT3 D835A (Nguyen et al, 2017) FLT3 D835G (Nguyen et al, 2017) FLT3 D835N (Nguyen et al, 2017) FLT3 D835Y (Nguyen et al, 2017)
Levis, M, Nguyen, B, Williams, AB, Small, D, Brown, P, Li, L, Young, DJ, Ma, H
Loss of function of tamatinib-resistant FLT3 mutants [plasma membrane]
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