The following FLT3 mutants are resistant to inhibition by sunitinib: FLT3 A848P (Albers et al, 2013) FLT3 D835A (Nguyen et al, 2017) FLT3 D835G (Nguyen et al, 2017) FLT3 D835N (Nguyen et al, 2017) FLT3 D835H (partial: Baker et al, 2013) FLT3 D835Y (partial: Baker et al, 2013; Nguyen et al, 2017) FLT3 D835A (Nguyen et al, 2017)
Yu, C, Albers, C, Verbeek, M, Duyster, J, Leischner, H, Illert, AL, von Bubnoff, N, Peschel, C
Loss of function of sunitinib-resistant FLT3 mutants [plasma membrane]
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