The following FLT3 mutants are resistant to inhibition by gilteritinib: FLT3 F691L (partial: Mori et al, 2017; Tarver et al, 2020) FLT3 F691I (partial: Mori et al, 2017)
Ueno, Y, Yamada, M, Kaneko, N, Kuromitsu, S, Mori, M, Saito, R, Shimada, I, Mori, K, Tanaka, R
Perl, AE, Mori, K, Hill, JE, Tarver, TC, Bahceci, E, Smith, CC, Rahmat, L
Loss of function of gilteritinib-resistant FLT3 mutants [plasma membrane]
© 2023 Reactome