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GHSR [plasma membrane]
Stable Identifier
R-HSA-947659
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
plasma membrane
Synonyms
Growth hormone secretagogue receptor type 1, GHSR_HUMAN
Locations in the PathwayBrowser
Expand all
Signal Transduction (Homo sapiens)
Signaling by GPCR (Homo sapiens)
GPCR downstream signalling (Homo sapiens)
G alpha (q) signalling events (Homo sapiens)
Liganded Gq-activating GPCRs bind inactive heterotrimeric Gq (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
Acyl ghrelin:GHSR [plasma membrane] (Homo sapiens)
GHSR [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
Acyl ghrelin:GHSR [plasma membrane] (Homo sapiens)
GHSR [plasma membrane] (Homo sapiens)
Liganded Gq/11-activating GPCRs act as GEFs for Gq/11 (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
Acyl ghrelin:GHSR [plasma membrane] (Homo sapiens)
GHSR [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
Acyl ghrelin:GHSR [plasma membrane] (Homo sapiens)
GHSR [plasma membrane] (Homo sapiens)
The Ligand:GPCR:Gq complex dissociates (Homo sapiens)
GPCRs that activate Gq/11 [plasma membrane] (Homo sapiens)
GHSR [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
Acyl ghrelin:GHSR [plasma membrane] (Homo sapiens)
GHSR [plasma membrane] (Homo sapiens)
GPCR ligand binding (Homo sapiens)
Class A/1 (Rhodopsin-like receptors) (Homo sapiens)
Peptide ligand-binding receptors (Homo sapiens)
GHSR is a receptor for ghrelin (Homo sapiens)
Acyl ghrelin:GHSR [plasma membrane] (Homo sapiens)
GHSR [plasma membrane] (Homo sapiens)
GHSR [plasma membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:Q92847 GHSR
Gene Names
GHSR
Chain
chain:1-366
Reference Genes
BioGPS Gene:2693 GHSR
COSMIC (genes):GHSR GHSR
CTD Gene:2693 GHSR
dbSNP Gene:2693 GHSR
ENSEMBL:ENSG00000121853 GHSR
HGNC:4267 GHSR
KEGG:hsa:2693 GHSR
Monarch:2693 GHSR
NCBI Gene:2693 GHSR
OMIM:601898 GHSR
UCSC:Q92847 GHSR
Reference Transcript
RefSeq:NM_004122.2 GHSR
RefSeq:NM_198407.2 GHSR
Participates
as an input of
GHSR is a receptor for ghrelin (Homo sapiens)
as a member of
GPCRs that activate Gq/11 [plasma membrane] (Homo sapiens)
as a component of
Acyl ghrelin:GHSR [plasma membrane] (Homo sapiens)
Inferred To
GHSR [plasma membrane]
(Bos taurus)
GHSR [plasma membrane]
(Canis familiaris)
GHSR [plasma membrane]
(Gallus gallus)
GHSR [plasma membrane]
(Sus scrofa)
PK2-R1 [plasma membrane]
(Drosophila melanogaster)
ghsr [plasma membrane]
(Xenopus tropicalis)
nmur-1 [plasma membrane]
(Caenorhabditis elegans)
nmur-2 [plasma membrane]
(Caenorhabditis elegans)
sphr-1 [plasma membrane]
(Caenorhabditis elegans)
Homologues of GHSR [plasma membrane]
(Caenorhabditis elegans)
Homologues of GHSR [plasma membrane]
(Drosophila melanogaster)
Homologues of GHSR [plasma membrane]
(Sus scrofa)
npr-20 [plasma membrane]
(Caenorhabditis elegans)
Ghsr [plasma membrane]
(Mus musculus)
Ghsr [plasma membrane]
(Rattus norvegicus)
PK1-R [plasma membrane]
(Drosophila melanogaster)
CapaR [plasma membrane]
(Drosophila melanogaster)
PK2-R2 [plasma membrane]
(Drosophila melanogaster)
Cross References
RefSeq
NP_940799.1
,
NP_004113.1
Guide to Pharmacology - Targets
246
ENSEMBL
ENSP00000395344
,
ENST00000427970
,
ENSG00000121853
,
ENST00000241256
,
ENSP00000241256
OpenTargets
ENSG00000121853
ZINC - Substances
GHSR_HUMAN
ZINC target
Q92847
PRO
Q92847
GlyGen
Q92847
PDB
6KO5
,
7NA8
,
7F9Z
,
7NA7
,
7F9Y
,
7W2Z
ZINC - Investigational
GHSR_HUMAN
GeneCards
GHSR
HPA
ENSG00000121853-GHSR
Pharos - Targets
Q92847
Orphanet
GHSR
ZINC - Predictions - Purchasable
GHSR_HUMAN
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