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RAPGEF1 [cytosol]
Stable Identifier
R-HSA-913472
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
cytosol
Synonyms
Rap guanine nucleotide exchange factor 1, RPGF1_HUMAN, C3G
Locations in the PathwayBrowser
Expand all
Immune System (Homo sapiens)
Cytokine Signaling in Immune system (Homo sapiens)
Signaling by Interleukins (Homo sapiens)
Interleukin-3, Interleukin-5 and GM-CSF signaling (Homo sapiens)
Regulation of signaling by CBL (Homo sapiens)
CBL:CRKL binds RAPGEF1 (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
p(Y700,731,774)-CBL:CRK:RAPGEF1 [cytosol] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
Signal Transduction (Homo sapiens)
Signaling by Erythropoietin (Homo sapiens)
Erythropoietin activates RAS (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1 binds SHC1 (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1 [plasma membrane] (Homo sapiens)
p-CRKL:RAPGEF1 [cytosol] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1:SHC1 [plasma membrane] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1 [plasma membrane] (Homo sapiens)
p-CRKL:RAPGEF1 [cytosol] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
EPO:p-EPOR:p-JAK2:LYN:IRS2 binds CRKL:RAPGEF1 (Homo sapiens)
CRKL:RAPGEF1 [cytosol] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:CRKL:RAPGEF1 [plasma membrane] (Homo sapiens)
CRKL:RAPGEF1 [cytosol] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
EPO:phospho-EPOR:phospho-JAK2:LYN:IRS2:phospho-CRKL:RAPGEF1:GRB2-1:SOS1,phospho-VAV1 mediates exchange of GTP for GDP bound to RAS (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1:p-Y-SHC1:GRB2:SOS1,p-Y-VAV1 [plasma membrane] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1:p-Y-SHC1:GRB2:SOS1 [plasma membrane] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1:p-Y-SHC1 [plasma membrane] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1 [plasma membrane] (Homo sapiens)
p-CRKL:RAPGEF1 [cytosol] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1:p-Y-SHC1:GRB2:p-Y-VAV1 [plasma membrane] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1:p-Y-SHC1 [plasma membrane] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1 [plasma membrane] (Homo sapiens)
p-CRKL:RAPGEF1 [cytosol] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
EPO:phospho-EPOR:phospho-JAK2:LYN:IRS2:phospho-CRKL:RAPGEF1:phospho-SHC1 binds GRB2:SOS1 (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1:p-Y-SHC1 [plasma membrane] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1 [plasma membrane] (Homo sapiens)
p-CRKL:RAPGEF1 [cytosol] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1:p-Y-SHC1:GRB2:SOS1 [plasma membrane] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1:p-Y-SHC1 [plasma membrane] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1 [plasma membrane] (Homo sapiens)
p-CRKL:RAPGEF1 [cytosol] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
EPO:phospho-EPOR:phospho-JAK2:LYN:IRS2:phospho-CRKL:RAPGEF1:phospho-SHC1 binds GRB2:VAV1 (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1:p-Y-SHC1 [plasma membrane] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1 [plasma membrane] (Homo sapiens)
p-CRKL:RAPGEF1 [cytosol] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1:p-Y-SHC1:GRB2:VAV1 [plasma membrane] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1:p-Y-SHC1 [plasma membrane] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1 [plasma membrane] (Homo sapiens)
p-CRKL:RAPGEF1 [cytosol] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
JAK2 phosphorylates SHC1 in EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:p-CRKL:RABGEF1:SHC1 (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1:SHC1 [plasma membrane] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1 [plasma membrane] (Homo sapiens)
p-CRKL:RAPGEF1 [cytosol] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1:p-Y-SHC1 [plasma membrane] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1 [plasma membrane] (Homo sapiens)
p-CRKL:RAPGEF1 [cytosol] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
JAK2 phosphorylates VAV1 in EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-Y-CRKL:RASGEF1:p-Y-SHC1:GRB2:VAV1 (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1:p-Y-SHC1:GRB2:VAV1 [plasma membrane] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1:p-Y-SHC1 [plasma membrane] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1 [plasma membrane] (Homo sapiens)
p-CRKL:RAPGEF1 [cytosol] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1:p-Y-SHC1:GRB2:p-Y-VAV1 [plasma membrane] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1:p-Y-SHC1 [plasma membrane] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1 [plasma membrane] (Homo sapiens)
p-CRKL:RAPGEF1 [cytosol] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
LYN phosphorylates CRKL in EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:CRKL:RAPGEF1 (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:CRKL:RAPGEF1 [plasma membrane] (Homo sapiens)
CRKL:RAPGEF1 [cytosol] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
EPO:p-8Y-EPOR:p-12Y-JAK2:LYN:IRS2:p-CRKL:RAPGEF1 [plasma membrane] (Homo sapiens)
p-CRKL:RAPGEF1 [cytosol] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
Signaling by Receptor Tyrosine Kinases (Homo sapiens)
Signaling by MET (Homo sapiens)
MET promotes cell motility (Homo sapiens)
MET activates RAP1 and RAC1 (Homo sapiens)
RAPGEF1 activates RAP1 (Homo sapiens)
HGF:p-4Y-MET:p-5Y-GAB1, HGF:p-4Y-MET:GRB2-1:p-5Y-GAB1:CRK,CRKL:RAPGEF1 [plasma membrane] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
RAPGEF1 binds CRK,CRKL (Homo sapiens)
HGF:p-4Y-MET:p-5Y-GAB1, HGF:p-4Y-MET:GRB2-1:p-5Y-GAB1:CRK,CRKL:RAPGEF1 [plasma membrane] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
Signaling by NTRKs (Homo sapiens)
Signaling by NTRK1 (TRKA) (Homo sapiens)
Signalling to ERKs (Homo sapiens)
Prolonged ERK activation events (Homo sapiens)
Frs2-mediated activation (Homo sapiens)
(Frs2)C3G stimulates nucleotide exchange on Rap1 (Homo sapiens)
Active TrkA receptor:p-FRS2:CRKL:RAPGEF1 [endosome membrane] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
p-FRS2:CRKL binds C3G (Homo sapiens)
Active TrkA receptor:p-FRS2:CRKL:RAPGEF1 [endosome membrane] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
RAPGEF1 [cytosol] (Homo sapiens)
External Reference Information
External Reference
UniProt:Q13905 RAPGEF1
Gene Names
RAPGEF1, GRF2
Chain
chain:1-1077
Reference Genes
BioGPS Gene:2889 RAPGEF1
COSMIC (genes):RAPGEF1 RAPGEF1
CTD Gene:2889 RAPGEF1
dbSNP Gene:2889 RAPGEF1
ENSEMBL:ENSG00000107263 RAPGEF1
HGNC:4568 RAPGEF1
KEGG Gene (Homo sapiens):2889 RAPGEF1
Monarch:2889 RAPGEF1
NCBI Gene:2889 RAPGEF1
OMIM:600303 RAPGEF1
UCSC:Q13905 RAPGEF1
Reference Transcript
RefSeq:NM_001304275.1 RAPGEF1
RefSeq:NM_005312.3 RAPGEF1
RefSeq:NM_198679.1 RAPGEF1
Other Identifiers
0003360215
0005220113
11716435_a_at
11742023_a_at
11748479_a_at
11756422_s_at
1570089_3p_at
1570089_at
17099208
204543_at
225738_at
226389_s_at
2889
3227689
3227690
3227691
3227692
3227693
3227694
3227695
3227697
3227698
3227702
3227704
3227706
3227708
3227710
3227711
3227712
3227713
3227714
3227722
3227732
3227735
3227738
3227757
3227761
3227762
3227763
3227764
3227765
3227766
3227767
3227772
3227773
3227778
3227780
3227802
3227813
3227814
3227815
36240_at
51157_at
65978_at
78805_at
8164665
A_23_P304237
A_23_P391764
D21239_at
GE543837
GE57112
GE79218
GE84667
GO:0000186
GO:0001568
GO:0002376
GO:0003674
GO:0005085
GO:0005515
GO:0005575
GO:0005622
GO:0005737
GO:0005768
GO:0005769
GO:0005829
GO:0006464
GO:0006810
GO:0006950
GO:0007155
GO:0007165
GO:0007169
GO:0007264
GO:0007267
GO:0007399
GO:0008150
GO:0008283
GO:0010976
GO:0016192
GO:0017034
GO:0017124
GO:0019221
GO:0019899
GO:0022607
GO:0030154
GO:0030670
GO:0031410
GO:0032486
GO:0032991
GO:0034330
GO:0038180
GO:0043226
GO:0043231
GO:0043547
GO:0046328
GO:0046579
GO:0046580
GO:0048008
GO:0048471
GO:0048856
GO:0051898
GO:0061028
GO:0070373
GO:0070374
GO:0071320
GO:0090090
GO:0090630
GO:0098609
GO:1901888
GO:1905451
GO:1990090
GO:2000178
Hs.9195.0.S1_3p_a_at
Hs.9195.1.S1_3p_x_at
Hs2.385815.1.S1_3p_at
Hs2.385815.1.S1_3p_x_at
ILMN_1769412
PH_hs_0022453
TC09001668.hg
g4885356_3p_at
Participant Of
hasComponent
Active TrkA receptor:p-FRS2:CRKL:RAPGEF1 [endosome membrane]
CRKL:RAPGEF1 [cytosol]
HGF:p-4Y-MET:p-5Y-GAB1, HGF:p-4Y-MET:GRB2-1:p-5Y-GAB1:CRK,CRKL:RAPGEF1 [plasma membrane]
p(Y700,731,774)-CBL:CRK:RAPGEF1 [cytosol]
p-CRKL:RAPGEF1 [cytosol]
input
CBL:CRKL binds RAPGEF1
p-FRS2:CRKL binds C3G
RAPGEF1 binds CRK,CRKL
Other forms of this molecule
RAPGEF1 [cytosol]
RAPGEF1 [endosome]
Inferred To
gbpD [cytosol] (Dictyostelium discoideum)
gefR [cytosol] (Dictyostelium discoideum)
gefA [cytosol] (Dictyostelium discoideum)
gefI [cytosol] (Dictyostelium discoideum)
gefJ [cytosol] (Dictyostelium discoideum)
Homologues of RAPGEF1 [cytosol] (Dictyostelium discoideum)
rapgef1b [cytosol] (Danio rerio)
gefH [cytosol] (Dictyostelium discoideum)
gefV [cytosol] (Dictyostelium discoideum)
Rapgef1 [cytosol] (Mus musculus)
Rapgef1 [cytosol] (Rattus norvegicus)
C3G [cytosol] (Drosophila melanogaster)
gefP [cytosol] (Dictyostelium discoideum)
gefF [cytosol] (Dictyostelium discoideum)
RAPGEF1 [cytosol] (Bos taurus)
RAPGEF1 [cytosol] (Caenorhabditis elegans)
RAPGEF1 [cytosol] (Canis familiaris)
RAPGEF1 [cytosol] (Dictyostelium discoideum)
RAPGEF1 [cytosol] (Gallus gallus)
RAPGEF1 [cytosol] (Sus scrofa)
RAPGEF1 [cytosol] (Xenopus tropicalis)
Cross References
RefSeq
NP_005303.2
,
NP_001291204.1
,
NP_941372.1
OpenTargets
ENSG00000107263
HPA
ENSG00000107263-RAPGEF1
GeneCards
Q13905
Ensembl
ENSP00000361264
,
ENST00000372189
,
ENSG00000107263
,
ENSP00000361269
,
ENST00000372190
,
ENST00000372195
,
ENSP00000361263
PRO
Q13905
PDB
5L23
Interactors (6)
Accession
#Entities
Entities
Confidence Score
Evidence (IntAct)
UniProt:P46108 CRK
1
CRK [cytosol]
(R-HSA-2980677)
0.758
6
UniProt:P62993 GRB2
1
GRB2 [cytosol]
(R-HSA-8983328)
0.658
3
UniProt:P00519 ABL1
5
p-Y226,Y393-ABL1 [nucleoplasm]
(R-HSA-8985251)
ABL1 [cytosol]
(R-HSA-375987)
p-S456-ABL1 [nucleoplasm]
(R-HSA-5686576)
ABL1 [nucleoplasm]
(R-HSA-5686579)
p-Y226,Y393-ABL1 [cytosol]
(R-HSA-8942610)
0.656
4
UniProt:P46109 CRKL
2
p-CRKL [cytosol]
(R-HSA-9024730)
CRKL [cytosol]
(R-HSA-354384)
0.641
3
UniProt:P46108-1 CRK
0.564
3
UniProt:P00533 EGFR
59
p-5Y-EGFRvIII [plasma membrane]
(R-HSA-1248649)
p-6Y-EGFR [clathrin-coated endocytic vesicle membrane]
(R-HSA-8869138)
EGFRvIII [plasma membrane]
(R-HSA-1214162)
p-6Y-EGFR E746_A750del;T790M [plasma membrane]
(R-HSA-1182985)
p-6Y-EGFR L858R;T790M [plasma membrane]
(R-HSA-1182984)
p-6Y-EGFR M766_A767insASV [plasma membrane]
(R-HSA-1996343)
p-6Y-EGFR D770_N771insNPH [plasma membrane]
(R-HSA-1996342)
p-6Y-EGFR V738_K739insKIPVAI [plasma membrane]
(R-HSA-1996346)
p-6Y-EGFR D770_N771insNPG [plasma membrane]
(R-HSA-1996335)
p-6Y-EGFR E746_A750del [plasma membrane]
(R-HSA-1181214)
p-6Y-EGFR L858R [plasma membrane]
(R-HSA-1173211)
p-6Y-EGFR G719S [plasma membrane]
(R-HSA-1169417)
p-6Y-EGFR L747_P753delinsS [plasma membrane]
(R-HSA-1228038)
p-6Y-EGFR L747_A750delinsP [plasma membrane]
(R-HSA-1228044)
p-6Y-EGFR L747_T751del [plasma membrane]
(R-HSA-1228041)
p-6Y-EGFR L747_S752del [plasma membrane]
(R-HSA-1228040)
p-6Y-EGFR L747_T751delinsP [plasma membrane]
(R-HSA-1228042)
p-6Y-EGFR E746_T751delinsA [plasma membrane]
(R-HSA-1228037)
p-6Y-EGFR E746_S752delinsV [plasma membrane]
(R-HSA-1228039)
p-6Y-EGFR L861Q [plasma membrane]
(R-HSA-1177541)
p-6Y-EGFR A289V [plasma membrane]
(R-HSA-1996334)
p-6Y-EGFR T263P [plasma membrane]
(R-HSA-1996336)
p-6Y-EGFR G598V [plasma membrane]
(R-HSA-1996339)
p-6Y-EGFR R108K [plasma membrane]
(R-HSA-1996338)
p-6Y-EGFR A289T [plasma membrane]
(R-HSA-1996341)
p-6Y-EGFR G719C [plasma membrane]
(R-HSA-1177530)
p-6Y-EGFR A289D [plasma membrane]
(R-HSA-1996340)
p-6Y-EGFR G719A [plasma membrane]
(R-HSA-1177528)
EGFR L858R;T790M [plasma membrane]
(R-HSA-1181386)
EGFR E746_A750del;T790M [plasma membrane]
(R-HSA-1181399)
EGFR D770_N771insNPG [plasma membrane]
(R-HSA-1996322)
EGFR V738_K739insKIPVAI [plasma membrane]
(R-HSA-1996325)
EGFR M766_A767insASV [plasma membrane]
(R-HSA-1996326)
EGFR D770_N771insNPH [plasma membrane]
(R-HSA-1996317)
EGFR L858R [plasma membrane]
(R-HSA-1173212)
EGFR G719S [plasma membrane]
(R-HSA-1169418)
EGFR E746_A750del [plasma membrane]
(R-HSA-1181211)
EGFR L747_P753delinsS [plasma membrane]
(R-HSA-1228010)
EGFR A289V [plasma membrane]
(R-HSA-1996321)
EGFR L747_T751delinsP [plasma membrane]
(R-HSA-1228012)
EGFR L747_T751del [plasma membrane]
(R-HSA-1228015)
EGFR A289D [plasma membrane]
(R-HSA-1996327)
EGFR L861Q [plasma membrane]
(R-HSA-1177542)
EGFR R108K [plasma membrane]
(R-HSA-1996330)
EGFR L747_A750delinsP [plasma membrane]
(R-HSA-1228034)
EGFR E746_T751delinsA [plasma membrane]
(R-HSA-1228031)
EGFR G719A [plasma membrane]
(R-HSA-1177532)
EGFR A289T [plasma membrane]
(R-HSA-1996306)
EGFR E746_S752delinsV [plasma membrane]
(R-HSA-1228025)
EGFR G719C [plasma membrane]
(R-HSA-1177531)
EGFR T263P [plasma membrane]
(R-HSA-1996315)
EGFR G598V [plasma membrane]
(R-HSA-1996314)
EGFR L747_S752del [plasma membrane]
(R-HSA-1228016)
EGFR [endosome membrane]
(R-HSA-9611160)
p-4Y-EGFR [plasma membrane]
(R-HSA-180287)
p-Y992,Y1045,Y1068,Y1086,Y1173-EGFR [plasma membrane]
(R-HSA-8864019)
p-Y1086,Y1101-EGFR [plasma membrane]
(R-HSA-179868)
EGFR [plasma membrane]
(R-HSA-179837)
p-6Y-EGFR [plasma membrane]
(R-HSA-179803)
0.553
2
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