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pS-ADRB2 [clathrin-coated endocytic vesicle membrane]
Stable Identifier
R-HSA-8869143
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
clathrin-coated endocytic vesicle membrane
Synonyms
Beta-2 adrenoceptor, RecName: Full=Beta-2 adrenergic receptor; AltName: Full=Beta-2 adrenoreceptor; Short=Beta-2 adrenoceptor;
GN Name=ADRB2; Synonyms=ADRB2R, B2AR;
OS Homo sapiens, ADRB2_HUMAN
Locations in the PathwayBrowser
Expand all
Vesicle-mediated transport (Homo sapiens)
Membrane Trafficking (Homo sapiens)
Clathrin-mediated endocytosis (Homo sapiens)
Auxilin recruits HSPA8:ATP to the clathrin-coated vesicle (Homo sapiens)
PI(4)P:p-T156 AP-2:clathrin:ITSNs:EPS15:REPS1:SGIP1:NECAPs:AAK1:CLASP proteins:cargo:F-BAR proteins:BAR domain proteins:ARP2/3 complex:WASL:f-actin:HIP dimers:DNM:GDP:SYNJs:auxilin [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
CLASP proteins:cargo [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB:ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2:Catecholamine [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2 [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
PI(4)P:p-T156 AP-2:clathrin:ITSNs:EPS15:REPS1:SGIP1:NECAPs:AAK1:CLASP proteins:cargo:F-BAR proteins:BAR domain proteins:ARP2/3 complex:WASL:f-actin:HIP dimers:DNM:GDP:SYNJs:auxilin:HSPA8:ATP [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
CLASP proteins:cargo [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB:ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2:Catecholamine [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2 [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
Clathrin recruits auxilins to the clathrin-coated vesicle (Homo sapiens)
PI(4)P:p-T156 AP-2:clathrin:ITSNs:EPS15:REPS1:SGIP1:NECAPs:AAK1:CLASP proteins:cargo:F-BAR proteins:BAR domain proteins:ARP2/3 complex:WASL:f-actin:HIP dimers:DNM:GDP:SYNJs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
CLASP proteins:cargo [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB:ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2:Catecholamine [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2 [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
PI(4)P:p-T156 AP-2:clathrin:ITSNs:EPS15:REPS1:SGIP1:NECAPs:AAK1:CLASP proteins:cargo:F-BAR proteins:BAR domain proteins:ARP2/3 complex:WASL:f-actin:HIP dimers:DNM:GDP:SYNJs:auxilin [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
CLASP proteins:cargo [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB:ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2:Catecholamine [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2 [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
Dissociation of AAK1 and dephosphorylation of AP-2 mu2 (Homo sapiens)
PI(4)P:p-T156 AP-2:ITSNs:EPS15:REPS1:SGIP1:NECAPs:AAK1:CLASP proteins:cargo:F-BAR proteins:BAR domain proteins:ARP2/3 complex:WASL:f-actin:HIP dimers:DNM:GDP:SYNJs:auxilin [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
PI(4)P:p-T156 AP-2:ITSNs:EPS15:REPS1:SGIP1:NECAPs:AAK1:CLASP proteins:cargo:F-BAR proteins:BAR domain proteins:ARP2/3 complex:WASL:f-actin:HIP dimers:DNM:GDP:SYNJs:auxilin [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
CLASP proteins:cargo [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB:ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2:Catecholamine [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2 [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
PI(4)P:p-T156 AP-2:ITSNs:EPS15:REPS1:SGIP1:NECAPs:CLASP proteins:cargo:F-BAR proteins:BAR domain proteins:ARP2/3 complex:WASL:f-actin:HIP dimers:DNM:GDP:SYNJs:auxilinGGC-RAB5:GTP:GAPVD1 [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
PI(4)P:ITSNs:EPS15:REPS1:NECAPs:AP-2:SGIP1:CLASP proteins:cargo:F-BAR proteins:BAR domain proteins:ARP2/3 complex:WASL:f-actin:HIP dimers:DNM:GDP:SYNJs:auxilin [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
CLASP proteins:cargo [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB:ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2:Catecholamine [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2 [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
Dissociation of clathrin-associated proteins (Homo sapiens)
CLASP proteins:cargo [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB:ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2:Catecholamine [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2 [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
PI(4)P:p-T156 AP-2:ITSNs:EPS15:REPS1:SGIP1:NECAPs:CLASP proteins:cargo:F-BAR proteins:BAR domain proteins:ARP2/3 complex:WASL:f-actin:HIP dimers:DNM:GDP:SYNJs:auxilinGGC-RAB5:GTP:GAPVD1 [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
PI(4)P:ITSNs:EPS15:REPS1:NECAPs:AP-2:SGIP1:CLASP proteins:cargo:F-BAR proteins:BAR domain proteins:ARP2/3 complex:WASL:f-actin:HIP dimers:DNM:GDP:SYNJs:auxilin [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
CLASP proteins:cargo [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB:ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2:Catecholamine [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2 [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
Dynamin-mediated GTP hydrolysis promotes vesicle scission (Homo sapiens)
PI(4)P:p-T156 AP-2:clathrin:ITSNs:EPS15:REPS1:SGIP1:NECAPs:AAK1:CLASP proteins:cargo:F-BAR proteins:BAR domain proteins:ARP2/3 complex:WASL:f-actin:HIP dimers:DNM:GDP:SYNJs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
CLASP proteins:cargo [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB:ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2:Catecholamine [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2 [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
HSPA8-mediated ATP hydrolysis promotes vesicle uncoating (Homo sapiens)
PI(4)P:p-T156 AP-2:ITSNs:EPS15:REPS1:SGIP1:NECAPs:AAK1:CLASP proteins:cargo:F-BAR proteins:BAR domain proteins:ARP2/3 complex:WASL:f-actin:HIP dimers:DNM:GDP:SYNJs:auxilin [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
CLASP proteins:cargo [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB:ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2:Catecholamine [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2 [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
PI(4)P:p-T156 AP-2:clathrin:ITSNs:EPS15:REPS1:SGIP1:NECAPs:AAK1:CLASP proteins:cargo:F-BAR proteins:BAR domain proteins:ARP2/3 complex:WASL:f-actin:HIP dimers:DNM:GDP:SYNJs:auxilin:HSPA8:ATP [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
CLASP proteins:cargo [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB:ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2:Catecholamine [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2 [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
RAB5 and GAPVD1 bind AP-2 (Homo sapiens)
PI(4)P:p-T156 AP-2:ITSNs:EPS15:REPS1:SGIP1:NECAPs:AAK1:CLASP proteins:cargo:F-BAR proteins:BAR domain proteins:ARP2/3 complex:WASL:f-actin:HIP dimers:DNM:GDP:SYNJs:auxilin [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
PI(4)P:p-T156 AP-2:ITSNs:EPS15:REPS1:SGIP1:NECAPs:AAK1:CLASP proteins:cargo:F-BAR proteins:BAR domain proteins:ARP2/3 complex:WASL:f-actin:HIP dimers:DNM:GDP:SYNJs:auxilin [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
CLASP proteins:cargo [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB:ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
ARRB-binding GPCRs [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2:Catecholamine [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
pS-ADRB2 [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:P07550 ADRB2
Gene Names
ADRB2, ADRB2R, B2AR
Chain
chain:1-413
Reference Genes
BioGPS Gene:154 ADRB2
COSMIC (genes):ADRB2 ADRB2
CTD Gene:154 ADRB2
dbSNP Gene:154 ADRB2
ENSEMBL:ENSG00000169252 ADRB2
HGNC:286 ADRB2
KEGG Gene (Homo sapiens):154 ADRB2
Monarch:154 ADRB2
NCBI Gene:154 ADRB2
Reference Transcript
RefSeq:NM_000024.5 ADRB2
Other Identifiers
0004590692
11728728_s_at
154
16990848
206170_PM_at
206170_at
2834747
2834748
2834749
2834750
2834751
2834752
2834753
2834754
2834755
610_at
8109086
A_14_P117388
A_14_P200154
A_23_P145024
GE80303
GO:0001540
GO:0001993
GO:0002024
GO:0002025
GO:0002028
GO:0002032
GO:0003013
GO:0003674
GO:0004930
GO:0004935
GO:0004941
GO:0005515
GO:0005575
GO:0005622
GO:0005634
GO:0005737
GO:0005764
GO:0005768
GO:0005769
GO:0005773
GO:0005794
GO:0005886
GO:0005887
GO:0006464
GO:0006810
GO:0006898
GO:0006914
GO:0006940
GO:0006950
GO:0007034
GO:0007165
GO:0007166
GO:0007171
GO:0007186
GO:0007188
GO:0007189
GO:0007190
GO:0007267
GO:0008150
GO:0008179
GO:0008333
GO:0009056
GO:0009058
GO:0009409
GO:0010008
GO:0010739
GO:0015459
GO:0016020
GO:0016021
GO:0016192
GO:0016324
GO:0019899
GO:0022607
GO:0030154
GO:0030501
GO:0030669
GO:0031410
GO:0031649
GO:0032991
GO:0034641
GO:0040007
GO:0040015
GO:0042592
GO:0042802
GO:0042803
GO:0043226
GO:0043235
GO:0043410
GO:0044877
GO:0045453
GO:0045944
GO:0045986
GO:0048856
GO:0050873
GO:0050877
GO:0051380
GO:0055085
GO:0061885
GO:0065003
GO:0071875
GO:0071880
GO:0071902
GO:0097746
GO:0120162
GO:1901098
GO:1904504
GO:1904646
GO:1990911
GO:2000481
GO:2000969
HMNXSV003031336
ILMN_1695590
J02960_cds1_s_at
M15169_at
PH_hs_0000339
TC05000814.hg
g13162366_3p_at
Participates
as a component of
pS-ADRB2:Catecholamine [clathrin-coated endocytic vesicle membrane] (Homo sapiens)
Other forms of this molecule
ADRB2 [endosome membrane]
PolyUb-ADRB2 [endosome membrane]
pS-ADRB2 [plasma membrane]
ADRB2 [plasma membrane]
Inferred To
Homologues of pS-ADRB2 [clathrin-coated endocytic vesicle membrane]
(Drosophila melanogaster)
phospho-adrb2 [clathrin-coated endocytic vesicle membrane]
(Xenopus tropicalis)
phospho-Octbeta3R [clathrin-coated endocytic vesicle membrane]
(Drosophila melanogaster)
phospho-DopEcR [clathrin-coated endocytic vesicle membrane]
(Drosophila melanogaster)
phospho-adrb2a [clathrin-coated endocytic vesicle membrane]
(Danio rerio)
phospho-ADRB2 [clathrin-coated endocytic vesicle membrane]
(Bos taurus)
phospho-ADRB2 [clathrin-coated endocytic vesicle membrane]
(Canis familiaris)
phospho-ADRB2 [clathrin-coated endocytic vesicle membrane]
(Sus scrofa)
phospho-Octbeta2R [clathrin-coated endocytic vesicle membrane]
(Drosophila melanogaster)
phospho-Octbeta1R [clathrin-coated endocytic vesicle membrane]
(Drosophila melanogaster)
phospho-Adrb2 [clathrin-coated endocytic vesicle membrane]
(Mus musculus)
phospho-Adrb2 [clathrin-coated endocytic vesicle membrane]
(Rattus norvegicus)
Modified Residues
Name
O-phospho-L-serine at unknown position
PsiMod Name
O-phospho-L-serine [MOD:00046]
PsiMod Definition
A protein modification that effectively converts an L-serine residue to O-phospho-L-serine.
Cross References
RefSeq
NP_000015.1
ZINC - World Drugs
ADRB2_HUMAN
Guide to Pharmacology - Targets
29
OpenTargets
ENSG00000169252
ZINC - FDA approved
ADRB2_HUMAN
ZINC - Substances
ADRB2_HUMAN
ZINC target
P07550
ZINC - Biogenic
ADRB2_HUMAN
PRO
P07550
PDB
6PS4
,
2R4S
,
6E67
,
3KJ6
,
3PDS
,
3P0G
,
6PS2
,
7BZ2
,
2R4R
,
6PS3
,
7DHR
,
5D5B
,
1GQ4
,
6KR8
,
5D5A
,
6PRZ
,
5JQH
,
6PS1
,
4LDO
,
6PS0
,
4LDL
,
5D6L
,
7DHI
,
6OBA
,
6NI3
,
3NYA
,
3NY9
,
4LDE
,
4GBR
,
4QKX
,
6N48
,
5X7D
,
3SN6
,
3D4S
,
3NY8
,
2RH1
,
6PS6
,
6PS5
,
6MXT
ZINC - Investigational
ADRB2_HUMAN
ZINC - Metabolites
ADRB2_HUMAN
GeneCards
P07550
HPA
ENSG00000169252-ADRB2
Ensembl
ENST00000305988
,
ENSG00000169252
,
ENSP00000305372
Pharos - Targets
P07550
Orphanet
27550
ZINC - Predictions - Purchasable
ADRB2_HUMAN
HMDB Protein
HMDBP01634
Interactors (30)
Accession
#Entities
Entities
Confidence Score
Evidence (IntAct)
UniProt:Q96B67 ARRD3
0.681
6
UniProt:P07550 ADRB2
5
pS-ADRB2 [clathrin-coated endocytic vesicle membrane]
(R-HSA-8869143)
ADRB2 [endosome membrane]
(R-HSA-6783036)
PolyUb-ADRB2 [endosome membrane]
(R-HSA-6783066)
pS-ADRB2 [plasma membrane]
(R-HSA-8852158)
ADRB2 [plasma membrane]
(R-HSA-390647)
0.657
4
UniProt:Q5TCQ9 MAGI3
0.619
9
UniProt:P63212 GNG2
1
GNG2 [plasma membrane]
(R-BTA-9717212)
0.612
4
UniProt:P54311 Gnb1
3
Gnb1 [photoreceptor disc membrane]
(R-RNO-55373)
G-protein beta 1 subunit [plasma membrane]
(R-RNO-421797)
Gnb1 [cytosol]
(R-RNO-6814412)
0.612
4
UniProt:P04896 GNAS2
0.612
4
UniProt:P12931 SRC
6
SRC [cytosol]
(R-HSA-9628701)
p-Y416-SRC [cytosol]
(R-HSA-8964276)
p-Y419-SRC [nucleoplasm]
(R-HSA-8937690)
MyrG-SRC [plasma membrane]
(R-HSA-8876922)
MyrG,p-Y530-SRC [plasma membrane]
(R-HSA-377598)
MyrG-p-Y419-SRC [plasma membrane]
(R-HSA-1810408)
0.611
3
UniProt:P30542 ADORA1
1
ADORA1 [plasma membrane]
(R-HSA-418941)
0.61
5
UniProt:P32121 ARRB2
2
ARRB2 [cytosol]
(R-HSA-416464)
PolyUb-ARRB2 [cytosol]
(R-HSA-6783000)
0.608
3
UniProt:O14745 NHRF1
0.558
6
UniProt:Q5T0J7-2 TEX35
0.556
3
UniProt:Q15910-2 EZH2
0.556
3
UniProt:O00472 ELL2
1
ELL2 [nucleoplasm]
(R-HSA-6807506)
0.556
3
UniProt:Q9H0X6 RN208
0.556
3
UniProt:Q9NR21-5 PARP11
0.556
3
UniProt:Q8WVD3 RNF138
1
RNF138 [cytosol]
(R-HSA-976008)
0.556
3
UniProt:A0AVK6 E2F8
1
E2F8 [nucleoplasm]
(R-HSA-8952990)
0.556
3
UniProt:Q5M9N0-2 CCDC158
0.556
3
UniProt:Q658K8 EF1DL
0.556
3
UniProt:Q13573 SNW1
1
SNW1 [nucleoplasm]
(R-HSA-351663)
0.556
3
UniProt:Q8N0U2 TMM61
0.556
3
UniProt:Q9UII2 ATIF1
0.556
3
UniProt:Q9NSI6-4 BRWD1
0.556
3
UniProt:Q15486 GUSP1
0.556
3
UniProt:Q9ULD4-2 Q9ULD42
0.556
3
UniProt:P61978 HNRNPK
2
polySUMO2-K422-HNRNPK [nucleoplasm]
(R-HSA-4570532)
HNRNPK [nucleoplasm]
(R-HSA-71945)
0.508
2
UniProt:Q99685 MGLL
3
MGLL [plasma membrane]
(R-HSA-426055)
MGLL [lipid droplet]
(R-HSA-163567)
MGLL [endoplasmic reticulum membrane]
(R-HSA-1500589)
0.508
2
UniProt:Q14232 EIF2B1
1
EIF2B1 [cytosol]
(R-HSA-72517)
0.463
2
UniProt:P04156 PRNP
2
PRNP [cytosol]
(R-HSA-9617597)
PRNP [plasma membrane]
(R-HSA-375060)
0.454
2
UniProt:P02686 MBP
1
MBP [cytosol]
(R-HSA-9614770)
0.454
2
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