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S-farn-GRK1 [photoreceptor disc membrane]
Stable Identifier
R-HSA-63140
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
photoreceptor disc membrane
Synonyms
S-fanesylated-Rhodopsin kinase
Locations in the PathwayBrowser
Expand all
Sensory Perception (Homo sapiens)
Visual phototransduction (Homo sapiens)
The phototransduction cascade (Homo sapiens)
Inactivation, recovery and regulation of the phototransduction cascade (Homo sapiens)
GRK1,4,7 phosphorylate MII to p-MII (Homo sapiens)
GRK1,4,7 [photoreceptor disc membrane] (Homo sapiens)
S-farn-GRK1 [photoreceptor disc membrane] (Homo sapiens)
S-farn-GRK1:RCVRN:Ca2+ [photoreceptor disc membrane] (Homo sapiens)
S-farn-GRK1 [photoreceptor disc membrane] (Homo sapiens)
RCVRN:Ca2+ binds to and inhibits GRK1 (Homo sapiens)
S-farn-GRK1 [photoreceptor disc membrane] (Homo sapiens)
S-farn-GRK1:RCVRN:Ca2+ [photoreceptor disc membrane] (Homo sapiens)
S-farn-GRK1 [photoreceptor disc membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:Q15835 GRK1
Gene Names
GRK1, RHOK
Chain
chain:1-560, propeptide:561-563
Reference Genes
BioGPS Gene:6011 GRK1
COSMIC (genes):GRK1 GRK1
CTD Gene:6011 GRK1
dbSNP Gene:6011 GRK1
ENSEMBL:ENSG00000185974 GRK1
HGNC:10013 GRK1
KEGG:hsa:6011 GRK1
Monarch:6011 GRK1
NCBI Gene:6011 GRK1
OMIM:180381 GRK1
UCSC:Q15835 GRK1
Reference Transcript
RefSeq:NM_002929.2 GRK1
Other Identifiers
11740741_a_at
11763482_at
16776924
208041_PM_at
208041_at
31562_at
3502804
3502805
3502806
3502808
3502810
6011
7970325
A_23_P313542
A_33_P3240867
GE579138
GE851521
GO:0001750
GO:0003824
GO:0004672
GO:0004674
GO:0004703
GO:0005524
GO:0005737
GO:0006468
GO:0007165
GO:0007601
GO:0008277
GO:0009966
GO:0016020
GO:0016056
GO:0016740
GO:0022400
GO:0042995
GO:0046777
GO:0050254
GO:0050877
GO:0097381
GO:0140096
HMNXSV003057502
ILMN_2216438
PH_hs_0035514
TC13000427.hg
g4506528_3p_at
Participates
as an input of
RCVRN:Ca2+ binds to and inhibits GRK1 (Homo sapiens)
as a component of
S-farn-GRK1:RCVRN:Ca2+ [photoreceptor disc membrane] (Homo sapiens)
as a member of
GRK1,4,7 [photoreceptor disc membrane] (Homo sapiens)
Inferred To
S-farn-GRK1 [photoreceptor disc membrane]
(Bos taurus)
S-farn-GRK1 [photoreceptor disc membrane]
(Caenorhabditis elegans)
S-farn-GRK1 [photoreceptor disc membrane]
(Danio rerio)
S-farn-GRK1 [photoreceptor disc membrane]
(Mus musculus)
S-farn-GRK1 [photoreceptor disc membrane]
(Rattus norvegicus)
S-farn-GRK1 [photoreceptor disc membrane]
(Sus scrofa)
GRK1 [photoreceptor disc membrane]
(Canis familiaris)
Modified Residues
Name
S-farnesyl-L-cysteine (farnesyl group) at 560
Coordinate
560
Modification
farnesyl group
PsiMod Name
S-farnesyl-L-cysteine [MOD:00111]
PsiMod Definition
A protein modification that effectively converts an L-cysteine residue to S-farnesyl-L-cysteine.
Cross References
ZINC - World Drugs
RK_HUMAN
Guide to Pharmacology - Targets
1465
ENSEMBL
ENST00000672946
,
ENST00000335678
,
ENSP00000499886
,
ENSP00000334876
OpenTargets
ENSG00000185974
ZINC - FDA approved
RK_HUMAN
ZINC - Substances
RK_HUMAN
ZINC - Biogenic
RK_HUMAN
ZINC target
Q15835
PRO
Q15835
PDB
5AFP
ZINC - Investigational
RK_HUMAN
HPA
ENSG00000185974-GRK1
Pharos - Targets
Q15835
Orphanet
GRK1
ZINC - Predictions - Purchasable
RK_HUMAN
HMDB Protein
HMDBP01418
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