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ADCYAP1R1 [plasma membrane]
Stable Identifier
R-HSA-420269
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
plasma membrane
Synonyms
Pituitary adenylate cyclase-activating polypeptide type I receptor, PACR_HUMAN
Locations in the PathwayBrowser
Expand all
Signal Transduction (Homo sapiens)
Signaling by GPCR (Homo sapiens)
GPCR downstream signalling (Homo sapiens)
G alpha (s) signalling events (Homo sapiens)
Liganded Gs-activating GPCR acts as a GEF for Gs (Homo sapiens)
GPCR:ligand complexes that act on Gs:Heterotrimeric G-protein Gs (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
ADCYAP1R1:ADCYAP1 peptides [plasma membrane] (Homo sapiens)
ADCYAP1R1 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs:Heterotrimeric G-protein Gs (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
ADCYAP1R1:ADCYAP1 peptides [plasma membrane] (Homo sapiens)
ADCYAP1R1 [plasma membrane] (Homo sapiens)
Liganded Gs-activating GPCRs bind inactive heterotrimeric Gs (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
ADCYAP1R1:ADCYAP1 peptides [plasma membrane] (Homo sapiens)
ADCYAP1R1 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs:Heterotrimeric G-protein Gs (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
ADCYAP1R1:ADCYAP1 peptides [plasma membrane] (Homo sapiens)
ADCYAP1R1 [plasma membrane] (Homo sapiens)
The Ligand:GPCR:Gs complex dissociates (Homo sapiens)
GPCR:ligand complexes that act on Gs:Heterotrimeric G-protein Gs (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
ADCYAP1R1:ADCYAP1 peptides [plasma membrane] (Homo sapiens)
ADCYAP1R1 [plasma membrane] (Homo sapiens)
GPCRs that activate Gs [plasma membrane] (Homo sapiens)
ADCYAP1R1 [plasma membrane] (Homo sapiens)
GPCR ligand binding (Homo sapiens)
Class B/2 (Secretin family receptors) (Homo sapiens)
Glucagon-type ligand receptors (Homo sapiens)
The PACAP receptor binds PACAP (Homo sapiens)
ADCYAP1R1 [plasma membrane] (Homo sapiens)
ADCYAP1R1:ADCYAP1 peptides [plasma membrane] (Homo sapiens)
ADCYAP1R1 [plasma membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:P41586 ADCYAP1R1
Gene Names
ADCYAP1R1
Chain
signal peptide:1-20, chain:21-468
Reference Genes
BioGPS Gene:117 ADCYAP1R1
COSMIC (genes):ADCYAP1R1 ADCYAP1R1
CTD Gene:117 ADCYAP1R1
dbSNP Gene:117 ADCYAP1R1
ENSEMBL:ENSG00000078549 ADCYAP1R1
HGNC:242 ADCYAP1R1
KEGG:hsa:117 ADCYAP1R1
Monarch:117 ADCYAP1R1
NCBI Gene:117 ADCYAP1R1
OMIM:102981 ADCYAP1R1
UCSC:P41586 ADCYAP1R1
Reference Transcript
RefSeq:XM_017011737.1 ADCYAP1R1
RefSeq:NM_001118.4 ADCYAP1R1
RefSeq:XM_005249618.4 ADCYAP1R1
RefSeq:NM_001199635.1 ADCYAP1R1
RefSeq:NM_001199637.1 ADCYAP1R1
RefSeq:NM_001199636.1 ADCYAP1R1
Participates
as an input of
The PACAP receptor binds PACAP (Homo sapiens)
as a member of
GPCRs that activate Gs [plasma membrane] (Homo sapiens)
as a component of
ADCYAP1R1:ADCYAP1 peptides [plasma membrane] (Homo sapiens)
Other forms of this molecule
ADCYAP1R1 [Golgi membrane]
Inferred To
ADCYAP1R1 [plasma membrane]
(Bos taurus)
ADCYAP1R1 [plasma membrane]
(Canis familiaris)
ADCYAP1R1 [plasma membrane]
(Gallus gallus)
ADCYAP1R1 [plasma membrane]
(Sus scrofa)
adcyap1r1a [plasma membrane]
(Danio rerio)
Adcyap1r1 [plasma membrane]
(Mus musculus)
Adcyap1r1 [plasma membrane]
(Rattus norvegicus)
Cross References
RefSeq
XP_016867226.1
,
NP_001186566.1
,
NP_001186565.1
,
XP_005249675.1
,
NP_001109.2
,
NP_001186564.1
Guide to Pharmacology - Targets
370
OpenTargets
ENSG00000078549
ENSEMBL
ENSP00000387335
,
ENST00000396211
,
ENSG00000078549
,
ENST00000705424
,
ENST00000409363
,
ENST00000304166
,
ENSP00000306620
,
ENSP00000379514
,
ENSP00000516125
ZINC - Substances
PACR_HUMAN
ZINC target
P41586
PRO
P41586
GlyGen
P41586
PDB
6LPB
,
8E3X
,
6P9Y
,
7JQD
,
3N94
,
2JOD
,
6M1I
,
6M1H
HPA
ENSG00000078549-ADCYAP1R1
GeneCards
ADCYAP1R1
Pharos - Targets
P41586
ZINC - Predictions - Purchasable
PACR_HUMAN
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