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CALCRL [plasma membrane]
Stable Identifier
R-HSA-419860
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
plasma membrane
Synonyms
Calcitonin gene-related peptide type 1 receptor, CALRL_HUMAN
Locations in the PathwayBrowser
Expand all
Signal Transduction (Homo sapiens)
Signaling by GPCR (Homo sapiens)
GPCR downstream signalling (Homo sapiens)
G alpha (s) signalling events (Homo sapiens)
Liganded Gs-activating GPCR acts as a GEF for Gs (Homo sapiens)
GPCR:ligand complexes that act on Gs:Heterotrimeric G-protein Gs (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
Adrenomedullin receptor:ADM,ADM2 [plasma membrane] (Homo sapiens)
Adrenomedullin receptor [plasma membrane] (Homo sapiens)
AM1 receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
AM2 receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
CGRP1 receptor:CGRP [plasma membrane] (Homo sapiens)
CGRP receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs:Heterotrimeric G-protein Gs (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
Adrenomedullin receptor:ADM,ADM2 [plasma membrane] (Homo sapiens)
Adrenomedullin receptor [plasma membrane] (Homo sapiens)
AM1 receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
AM2 receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
CGRP1 receptor:CGRP [plasma membrane] (Homo sapiens)
CGRP receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
Liganded Gs-activating GPCRs bind inactive heterotrimeric Gs (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
Adrenomedullin receptor:ADM,ADM2 [plasma membrane] (Homo sapiens)
Adrenomedullin receptor [plasma membrane] (Homo sapiens)
AM1 receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
AM2 receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
CGRP1 receptor:CGRP [plasma membrane] (Homo sapiens)
CGRP receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs:Heterotrimeric G-protein Gs (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
Adrenomedullin receptor:ADM,ADM2 [plasma membrane] (Homo sapiens)
Adrenomedullin receptor [plasma membrane] (Homo sapiens)
AM1 receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
AM2 receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
CGRP1 receptor:CGRP [plasma membrane] (Homo sapiens)
CGRP receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
The Ligand:GPCR:Gs complex dissociates (Homo sapiens)
GPCR:ligand complexes that act on Gs:Heterotrimeric G-protein Gs (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
Adrenomedullin receptor:ADM,ADM2 [plasma membrane] (Homo sapiens)
Adrenomedullin receptor [plasma membrane] (Homo sapiens)
AM1 receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
AM2 receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
CGRP1 receptor:CGRP [plasma membrane] (Homo sapiens)
CGRP receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
GPCRs that activate Gs [plasma membrane] (Homo sapiens)
Adrenomedullin receptor [plasma membrane] (Homo sapiens)
AM1 receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
AM2 receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
CGRP receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
GPCR ligand binding (Homo sapiens)
Class B/2 (Secretin family receptors) (Homo sapiens)
Calcitonin-like ligand receptors (Homo sapiens)
CGRP receptor can bind calcitonin gene-related peptides (Homo sapiens)
CGRP receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
CGRP1 receptor:CGRP [plasma membrane] (Homo sapiens)
CGRP receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
The adrenomedullin receptor can bind adrenomedullin and intermedin (Homo sapiens)
Adrenomedullin receptor [plasma membrane] (Homo sapiens)
AM1 receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
AM2 receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
Adrenomedullin receptor:ADM,ADM2 [plasma membrane] (Homo sapiens)
Adrenomedullin receptor [plasma membrane] (Homo sapiens)
AM1 receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
AM2 receptor [plasma membrane] (Homo sapiens)
CALCRL [plasma membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:Q16602 CALCRL
Gene Names
CALCRL, CGRPR
Chain
signal peptide:1-22, chain:23-461
Reference Genes
BioGPS Gene:10203 CALCRL
COSMIC (genes):CALCRL CALCRL
CTD Gene:10203 CALCRL
dbSNP Gene:10203 CALCRL
ENSEMBL:ENSG00000064989 CALCRL
ENSEMBL:ENSG00000064989.13 CALCRL
HGNC:16709 CALCRL
KEGG Gene (Homo sapiens):10203 CALCRL
Monarch:10203 CALCRL
NCBI Gene:10203 CALCRL
OMIM:114190 CALCRL
UCSC:Q16602 CALCRL
Reference Transcript
RefSeq:NM_001271751.1 CALCRL
RefSeq:NM_005795.5 CALCRL
Other Identifiers
10203
11730274_at
11730275_at
11747993_a_at
16906285
206331_PM_at
206331_at
210815_PM_s_at
210815_s_at
234996_PM_at
234996_at
2591366
2591368
2591369
2591370
2591371
2591372
2591373
2591374
2591375
2591376
2591378
2591379
2591381
2591383
2591384
2591385
2591386
2591388
2591389
2591390
2591399
2591402
34995_at
42475_at
59645_at
8057578
A_23_P39898
A_33_P3261957
A_33_P3306103
A_33_P3306110
GE57788
GO:0001525
GO:0001605
GO:0001635
GO:0004888
GO:0004930
GO:0004948
GO:0005515
GO:0005737
GO:0005764
GO:0005768
GO:0005773
GO:0005783
GO:0005886
GO:0006816
GO:0007165
GO:0007166
GO:0007186
GO:0007187
GO:0007189
GO:0007507
GO:0008283
GO:0008284
GO:0015031
GO:0016020
GO:0016192
GO:0023052
GO:0031410
GO:0031623
GO:0043226
GO:0048659
GO:0048856
GO:0060089
GO:0071329
GO:1903143
GO:1904707
GO:1990406
GO:1990408
GO:1990409
GO:1990410
GO:1990874
HMNXSV003028892
Hs.201591.0.A1_3p_at
ILMN_1758281
L76380_at
TC02002605.hg
g5031620_3p_x_at
g662328_3p_a_at
Participates
as a component of
AM1 receptor [plasma membrane] (Homo sapiens)
AM2 receptor [plasma membrane] (Homo sapiens)
CGRP receptor [plasma membrane] (Homo sapiens)
Inferred To
CALCRL [plasma membrane]
(Bos taurus)
CALCRL [plasma membrane]
(Canis familiaris)
CALCRL [plasma membrane]
(Gallus gallus)
CALCRL [plasma membrane]
(Sus scrofa)
Calcrl [plasma membrane]
(Mus musculus)
Calcrl [plasma membrane]
(Rattus norvegicus)
calcrla [plasma membrane]
(Danio rerio)
calcrl [plasma membrane]
(Xenopus tropicalis)
Cross References
RefSeq
NP_005786.1
,
NP_001258680.1
Guide to Pharmacology - Targets
47
OpenTargets
ENSG00000064989
ZINC - Substances
CALRL_HUMAN
ZINC target
Q16602
PRO
Q16602
PDB
3N7R
,
3N7P
,
6D1U
,
6UUS
,
6UVA
,
7KNT
,
8AX5
,
7P0F
,
8AX6
,
6ZHO
,
6UUN
,
6UMG
,
7P0I
,
8AX7
,
7KNU
,
4RWG
,
6V2E
,
3N7S
,
5V6Y
,
6ZIS
,
6E3Y
,
4RWF
,
3AQF
ZINC - Investigational
CALRL_HUMAN
HPA
ENSG00000064989-CALCRL
GeneCards
Q16602
Ensembl
ENST00000409998
,
ENSP00000376177
,
ENST00000392370
,
ENSG00000064989
,
ENST00000410068
,
ENSP00000386972
,
ENSP00000387190
Pharos - Targets
Q16602
ZINC - Predictions - Purchasable
CALRL_HUMAN
HMDB Protein
HMDBP13628
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