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CALCR [plasma membrane]
Stable Identifier
R-HSA-419798
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
plasma membrane
Synonyms
Calcitonin receptor, CALCR_HUMAN
Locations in the PathwayBrowser
Expand all
Signal Transduction (Homo sapiens)
Signaling by GPCR (Homo sapiens)
GPCR downstream signalling (Homo sapiens)
G alpha (s) signalling events (Homo sapiens)
Liganded Gs-activating GPCR acts as a GEF for Gs (Homo sapiens)
GPCR:ligand complexes that act on Gs:Heterotrimeric G-protein Gs (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
AMY1-3:IAPP(34-70) [plasma membrane] (Homo sapiens)
AMY1-3 [plasma membrane] (Homo sapiens)
AMY1 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
AMY2 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
AMY3 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
CALCR:CALCA(83-119) [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs:Heterotrimeric G-protein Gs (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
AMY1-3:IAPP(34-70) [plasma membrane] (Homo sapiens)
AMY1-3 [plasma membrane] (Homo sapiens)
AMY1 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
AMY2 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
AMY3 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
CALCR:CALCA(83-119) [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
Liganded Gs-activating GPCRs bind inactive heterotrimeric Gs (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
AMY1-3:IAPP(34-70) [plasma membrane] (Homo sapiens)
AMY1-3 [plasma membrane] (Homo sapiens)
AMY1 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
AMY2 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
AMY3 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
CALCR:CALCA(83-119) [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs:Heterotrimeric G-protein Gs (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
AMY1-3:IAPP(34-70) [plasma membrane] (Homo sapiens)
AMY1-3 [plasma membrane] (Homo sapiens)
AMY1 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
AMY2 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
AMY3 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
CALCR:CALCA(83-119) [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
The Ligand:GPCR:Gs complex dissociates (Homo sapiens)
GPCR:ligand complexes that act on Gs:Heterotrimeric G-protein Gs (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
AMY1-3:IAPP(34-70) [plasma membrane] (Homo sapiens)
AMY1-3 [plasma membrane] (Homo sapiens)
AMY1 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
AMY2 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
AMY3 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
CALCR:CALCA(83-119) [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
GPCRs that activate Gs [plasma membrane] (Homo sapiens)
AMY1-3 [plasma membrane] (Homo sapiens)
AMY1 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
AMY2 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
AMY3 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
GPCR ligand binding (Homo sapiens)
Class B/2 (Secretin family receptors) (Homo sapiens)
Calcitonin-like ligand receptors (Homo sapiens)
AMY1-3 bind IAPP(34-70) (Homo sapiens)
AMY1-3 [plasma membrane] (Homo sapiens)
AMY1 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
AMY2 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
AMY3 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
AMY1-3:IAPP(34-70) [plasma membrane] (Homo sapiens)
AMY1-3 [plasma membrane] (Homo sapiens)
AMY1 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
AMY2 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
AMY3 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
AMY1-3 bind pramlintide (Homo sapiens)
AMY1-3 [plasma membrane] (Homo sapiens)
AMY1 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
AMY2 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
AMY3 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
AMY1-3:pramlintide [plasma membrane] (Homo sapiens)
AMY1-3 [plasma membrane] (Homo sapiens)
AMY1 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
AMY2 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
AMY3 receptor [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
CALCA(83-119) binds CALCR (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
CALCR:CALCA(83-119) [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
CALCR binds erenumab (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
CALCR:erenumab [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
CALCR binds gepants (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
CALCR:gepants [plasma membrane] (Homo sapiens)
CALCR [plasma membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:P30988 CALCR
Gene Names
CALCR
Chain
signal peptide:1-24, chain:25-474
Reference Genes
BioGPS Gene:799 CALCR
COSMIC (genes):CALCR CALCR
CTD Gene:799 CALCR
dbSNP Gene:799 CALCR
ENSEMBL:ENSG00000004948 CALCR
HGNC:1440 CALCR
KEGG:hsa:799 CALCR
Monarch:799 CALCR
NCBI Gene:799 CALCR
OMIM:114131 CALCR
UCSC:P30988 CALCR
Reference Transcript
RefSeq:NM_001742.3 CALCR
RefSeq:NM_001164738.1 CALCR
RefSeq:NM_001164737.1 CALCR
Other Identifiers
11736980_a_at
11736981_a_at
17059804
207886_PM_s_at
207886_s_at
207887_PM_s_at
207887_s_at
3061539
3061540
3061541
3061542
3061545
3061546
3061547
3061548
3061550
3061553
3061554
3061555
3061556
3061557
3061558
3061559
3061561
3061562
3061564
3061573
3061574
3061579
3061580
36746_s_at
799
8140995
A_23_P134484
A_33_P3710082
GE80667
GO:0001503
GO:0001540
GO:0001635
GO:0001669
GO:0004888
GO:0004930
GO:0004948
GO:0005515
GO:0005886
GO:0005929
GO:0007166
GO:0007186
GO:0007188
GO:0007189
GO:0007204
GO:0010628
GO:0010739
GO:0016020
GO:0030154
GO:0030279
GO:0030316
GO:0030424
GO:0031410
GO:0032841
GO:0043226
GO:0043488
GO:0050850
GO:0051384
GO:0051897
GO:0060089
GO:0070374
GO:0097643
GO:0097647
GO:0150056
GO:0150057
GO:0150058
GO:1904645
GO:1990408
HMNXSV003023985
ILMN_1710219
PH_hs_0000072
TC07001608.hg
X69920_s_at
g4502546_3p_a_at
g6456429_3p_a_at
Participates
as a component of
CALCR:erenumab [plasma membrane] (Homo sapiens)
CALCR:gepants [plasma membrane] (Homo sapiens)
AMY2 receptor [plasma membrane] (Homo sapiens)
AMY3 receptor [plasma membrane] (Homo sapiens)
AMY1 receptor [plasma membrane] (Homo sapiens)
CALCR:CALCA(83-119) [plasma membrane] (Homo sapiens)
as an input of
CALCR binds erenumab (Homo sapiens)
CALCR binds gepants (Homo sapiens)
CALCA(83-119) binds CALCR (Homo sapiens)
as a member of
GPCRs that activate Gs [plasma membrane] (Homo sapiens)
Inferred To
CALCR [plasma membrane]
(Bos taurus)
CALCR [plasma membrane]
(Canis familiaris)
CALCR [plasma membrane]
(Gallus gallus)
CALCR [plasma membrane]
(Sus scrofa)
calcr [plasma membrane]
(Xenopus tropicalis)
Calcr [plasma membrane]
(Mus musculus)
Calcr [plasma membrane]
(Rattus norvegicus)
hec [plasma membrane]
(Drosophila melanogaster)
seb-2 [plasma membrane]
(Caenorhabditis elegans)
Dh31-R [plasma membrane]
(Drosophila melanogaster)
Homologues of CALCR [plasma membrane]
(Drosophila melanogaster)
Cross References
RefSeq
NP_001158209.1
,
NP_001733.1
,
NP_001158210.1
Guide to Pharmacology - Targets
43
OpenTargets
ENSG00000004948
ENSEMBL
ENSP00000377959
,
ENSP00000389295
,
ENST00000415529
,
ENST00000426151
,
ENSP00000413179
,
ENST00000423724
,
ENSP00000391369
,
ENSP00000497687
,
ENST00000394441
,
ENST00000649521
ZINC - Substances
CALCR_HUMAN
ZINC target
P30988
PRO
P30988
Pharos - Targets
P30988
GlyGen
P30988
ZINC - Predictions - Purchasable
CALCR_HUMAN
PDB
7TYI
,
5II0
,
7TYW
,
7TYO
,
7TYN
,
7TYL
,
9AUC
,
8F2B
,
6PGQ
,
8F2A
,
6PFO
,
6NIY
,
8F0J
,
7TYF
,
7TZF
,
7TYY
,
8F0K
,
5UZ7
,
7TYX
,
7TYH
HMDB Protein
HMDBP12709
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