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HTR1E [plasma membrane]
Stable Identifier
R-HSA-390960
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
plasma membrane
Synonyms
5-HT1E receptor, RecName: Full=5-hydroxytryptamine receptor 1E; Short=5-HT-1E; Short=5-HT1E; AltName: Full=Serotonin receptor 1E; AltName: Full=S31;
GN Name=HTR1E;
OS Homo sapiens, 5HT1E_HUMAN
Locations in the PathwayBrowser
Expand all
Signal Transduction (Homo sapiens)
Signaling by GPCR (Homo sapiens)
GPCR downstream signalling (Homo sapiens)
G alpha (i) signalling events (Homo sapiens)
Liganded Gi-activating GPCR acts as a GEF for Gi (Homo sapiens)
Ligand:GPCR complexes that activate Gi:Heterotrimeric G-protein Gi (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
HTR1B,D,E,F,HTR5A:5HT [plasma membrane] (Homo sapiens)
HTR1B,D,E,F,HTR5A [plasma membrane] (Homo sapiens)
HTR1E [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi:Heterotrimeric G-protein Gi (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
HTR1B,D,E,F,HTR5A:5HT [plasma membrane] (Homo sapiens)
HTR1B,D,E,F,HTR5A [plasma membrane] (Homo sapiens)
HTR1E [plasma membrane] (Homo sapiens)
Liganded Gi-activating GPCRs bind inactive heterotrimeric G-protein Gi (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
HTR1B,D,E,F,HTR5A:5HT [plasma membrane] (Homo sapiens)
HTR1B,D,E,F,HTR5A [plasma membrane] (Homo sapiens)
HTR1E [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi:Heterotrimeric G-protein Gi (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
HTR1B,D,E,F,HTR5A:5HT [plasma membrane] (Homo sapiens)
HTR1B,D,E,F,HTR5A [plasma membrane] (Homo sapiens)
HTR1E [plasma membrane] (Homo sapiens)
The Ligand:GPCR:Gi complex dissociates (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
HTR1B,D,E,F,HTR5A:5HT [plasma membrane] (Homo sapiens)
HTR1B,D,E,F,HTR5A [plasma membrane] (Homo sapiens)
HTR1E [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi:Heterotrimeric G-protein Gi (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
HTR1B,D,E,F,HTR5A:5HT [plasma membrane] (Homo sapiens)
HTR1B,D,E,F,HTR5A [plasma membrane] (Homo sapiens)
HTR1E [plasma membrane] (Homo sapiens)
GPCR ligand binding (Homo sapiens)
Class A/1 (Rhodopsin-like receptors) (Homo sapiens)
Amine ligand-binding receptors (Homo sapiens)
Serotonin receptors (Homo sapiens)
HTR1 and 5A receptors can bind serotonin (Homo sapiens)
HTR1B,D,E,F,HTR5A [plasma membrane] (Homo sapiens)
HTR1E [plasma membrane] (Homo sapiens)
HTR1B,D,E,F,HTR5A:5HT [plasma membrane] (Homo sapiens)
HTR1B,D,E,F,HTR5A [plasma membrane] (Homo sapiens)
HTR1E [plasma membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:P28566 HTR1E
Gene Names
HTR1E
Chain
chain:1-365
Reference Genes
BioGPS Gene:3354 HTR1E
COSMIC (genes):HTR1E HTR1E
CTD Gene:3354 HTR1E
dbSNP Gene:3354 HTR1E
ENSEMBL:ENSG00000168830 HTR1E
ENSEMBL:ENSG00000168830.8 HTR1E
HGNC:5291 HTR1E
KEGG Gene (Homo sapiens):3354 HTR1E
Monarch:3354 HTR1E
NCBI Gene:3354 HTR1E
OMIM:182132 HTR1E
UCSC:P28566 HTR1E
Reference Transcript
RefSeq:NM_000865.2 HTR1E
RefSeq:XM_011535789.2 HTR1E
Other Identifiers
11752511_a_at
17010782
207404_PM_s_at
207404_s_at
2916075
2916076
2916077
2916078
2916094
2916095
2916096
2916097
2916098
2916099
2916100
2916101
2916102
2916103
3354
33607_at
8120983
A_14_P112758
A_23_P70648
A_24_P380349
GE58138
GO:0004930
GO:0004993
GO:0005515
GO:0005886
GO:0007165
GO:0007186
GO:0007187
GO:0007193
GO:0007198
GO:0007268
GO:0016020
GO:0023052
GO:0030425
GO:0030594
GO:0045202
GO:0051378
GO:0060089
HMNXSV003032387
ILMN_1794095
M91467_at
PH_hs_0000220
TC06000782.hg
TC06002912.hg
g4504536_3p_a_at
Participates
as a member of
HTR1B,D,E,F,HTR5A [plasma membrane] (Homo sapiens)
Inferred To
octr-1 [plasma membrane]
(Caenorhabditis elegans)
HTR1E [plasma membrane]
(Bos taurus)
HTR1E [plasma membrane]
(Gallus gallus)
HTR1E [plasma membrane]
(Sus scrofa)
htr1e [plasma membrane]
(Xenopus tropicalis)
Cross References
RefSeq
XP_011534091.1
,
NP_000856.1
ZINC - World Drugs
5HT1E_HUMAN
Guide to Pharmacology - Targets
4
OpenTargets
ENSG00000168830
ZINC - FDA approved
5HT1E_HUMAN
ZINC - Substances
5HT1E_HUMAN
ZINC - Biogenic
5HT1E_HUMAN
ZINC target
P28566
PRO
P28566
PDB
7E33
ZINC - Investigational
5HT1E_HUMAN
ZINC - Metabolites
5HT1E_HUMAN
GeneCards
P28566
HPA
ENSG00000168830-HTR1E
Ensembl
ENSP00000307766
,
ENSG00000168830
,
ENST00000305344
Pharos - Targets
P28566
ZINC - Predictions - Purchasable
5HT1E_HUMAN
HMDB Protein
HMDBP10858
Interactors (1)
Accession
#Entities
Entities
Confidence Score
Evidence (IntAct)
UniProt:Q96CV9 OPTN
5
OPTN [recycling endosome membrane]
(R-HSA-8854141)
p-S177-OPTN [nucleoplasm]
(R-HSA-2562595)
p-S177-OPTN [cytosol]
(R-HSA-2562525)
OPTN [Golgi membrane]
(R-HSA-2161111)
OPTN [cytosol]
(R-HSA-9687907)
0.556
3
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