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HTR2A [plasma membrane]
Stable Identifier
R-HSA-390947
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
plasma membrane
Synonyms
5-HT2A receptor, RecName: Full=5-hydroxytryptamine receptor 2A; Short=5-HT-2A; Short=5-HT-2; AltName: Full=Serotonin receptor 2A;
GN Name=HTR2A; Synonyms=HTR2;
OS Homo sapiens, 5HT2A_HUMAN
Icon
Locations in the PathwayBrowser
Expand all
Signal Transduction (Homo sapiens)
Signaling by GPCR (Homo sapiens)
GPCR downstream signalling (Homo sapiens)
G alpha (q) signalling events (Homo sapiens)
Liganded Gq-activating GPCRs bind inactive heterotrimeric Gq (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
HTR2A-C:5HT [plasma membrane] (Homo sapiens)
HTR2A-C [plasma membrane] (Homo sapiens)
HTR2A [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
HTR2A-C:5HT [plasma membrane] (Homo sapiens)
HTR2A-C [plasma membrane] (Homo sapiens)
HTR2A [plasma membrane] (Homo sapiens)
Liganded Gq/11-activating GPCRs act as GEFs for Gq/11 (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
HTR2A-C:5HT [plasma membrane] (Homo sapiens)
HTR2A-C [plasma membrane] (Homo sapiens)
HTR2A [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
HTR2A-C:5HT [plasma membrane] (Homo sapiens)
HTR2A-C [plasma membrane] (Homo sapiens)
HTR2A [plasma membrane] (Homo sapiens)
The Ligand:GPCR:Gq complex dissociates (Homo sapiens)
GPCRs that activate Gq/11 [plasma membrane] (Homo sapiens)
HTR2A-C [plasma membrane] (Homo sapiens)
HTR2A [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
HTR2A-C:5HT [plasma membrane] (Homo sapiens)
HTR2A-C [plasma membrane] (Homo sapiens)
HTR2A [plasma membrane] (Homo sapiens)
GPCR ligand binding (Homo sapiens)
Class A/1 (Rhodopsin-like receptors) (Homo sapiens)
Amine ligand-binding receptors (Homo sapiens)
Serotonin receptors (Homo sapiens)
5-HT2 receptor can bind serotonin (Homo sapiens)
HTR2A-C [plasma membrane] (Homo sapiens)
HTR2A [plasma membrane] (Homo sapiens)
HTR2A-C:5HT [plasma membrane] (Homo sapiens)
HTR2A-C [plasma membrane] (Homo sapiens)
HTR2A [plasma membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:P28223 HTR2A
Gene Names
HTR2A, HTR2
Chain
chain:1-471
Reference Genes
BioGPS Gene:3356 HTR2A
COSMIC (genes):HTR2A HTR2A
CTD Gene:3356 HTR2A
dbSNP Gene:3356 HTR2A
ENSEMBL:ENSG00000102468.11 HTR2A
HGNC:5293 HTR2A
KEGG Gene (Homo sapiens):3356 HTR2A
Monarch:3356 HTR2A
NCBI Gene:3356 HTR2A
OMIM:182135 HTR2A
UCSC:P28223 HTR2A
Reference Transcript
RefSeq:NM_001165947.2 HTR2A
RefSeq:NM_000621.4 HTR2A
Other Identifiers
11736750_a_at
11736751_at
11736752_x_at
11750398_a_at
16778938
207135_PM_at
207135_at
211616_PM_s_at
211616_s_at
244130_PM_at
244130_at
3356
3513146
3513149
3513150
3513151
3513152
3513174
3513176
3513177
3513178
3513180
3513208
3513210
3513212
35469_at
35471_g_at
60209_at
7971526
A_24_P355967
GE588095
GE59830
GO:0001587
GO:0001618
GO:0001659
GO:0003012
GO:0003013
GO:0004930
GO:0004993
GO:0005515
GO:0005737
GO:0005829
GO:0005886
GO:0005887
GO:0005901
GO:0005975
GO:0006091
GO:0006096
GO:0006629
GO:0006874
GO:0007165
GO:0007186
GO:0007187
GO:0007200
GO:0007202
GO:0007204
GO:0007208
GO:0007210
GO:0007268
GO:0007568
GO:0007610
GO:0007613
GO:0008219
GO:0008284
GO:0009410
GO:0010513
GO:0014059
GO:0014065
GO:0014824
GO:0014832
GO:0016020
GO:0016021
GO:0018108
GO:0019233
GO:0023052
GO:0030154
GO:0030424
GO:0030425
GO:0030431
GO:0030594
GO:0031410
GO:0033674
GO:0036211
GO:0042734
GO:0042802
GO:0042995
GO:0043025
GO:0043198
GO:0043226
GO:0043267
GO:0043406
GO:0044380
GO:0044877
GO:0045202
GO:0045211
GO:0045600
GO:0045821
GO:0045907
GO:0046718
GO:0048148
GO:0050731
GO:0050877
GO:0050965
GO:0050966
GO:0051209
GO:0051378
GO:0051967
GO:0055065
GO:0055085
GO:0055086
GO:0060089
GO:0070374
GO:0070852
GO:0071886
GO:0098664
GO:0098666
GO:0098793
GO:0098978
GO:0099171
GO:1901135
HMNXSV003042038
Hs.72630.0.A1_3p_at
ILMN_1715496
PH_hs_0025180
TC13000648.hg
TC13001479.hg
X57830_at
g10835174_3p_at
g177775_3p_s_at
Participates
as a member of
HTR2A-C [plasma membrane] (Homo sapiens)
Inferred To
Homologues of HTR2A [plasma membrane]
(Caenorhabditis elegans)
5-HT2B [plasma membrane]
(Drosophila melanogaster)
htr2a [plasma membrane]
(Xenopus tropicalis)
HTR2A [plasma membrane]
(Bos taurus)
HTR2A [plasma membrane]
(Canis familiaris)
HTR2A [plasma membrane]
(Danio rerio)
HTR2A [plasma membrane]
(Gallus gallus)
HTR2A [plasma membrane]
(Mus musculus)
HTR2A [plasma membrane]
(Rattus norvegicus)
HTR2A [plasma membrane]
(Sus scrofa)
dop-6 [plasma membrane]
(Caenorhabditis elegans)
tag-89 [plasma membrane]
(Caenorhabditis elegans)
Cross References
RefSeq
NP_000612.1
,
NP_001159419.1
ZINC - World Drugs
5HT2A_HUMAN
Guide to Pharmacology - Targets
6
OpenTargets
ENSG00000102468
ZINC - FDA approved
5HT2A_HUMAN
ZINC - Substances
5HT2A_HUMAN
ZINC target
P28223
ZINC - Biogenic
5HT2A_HUMAN
PRO
P28223
PDB
6A93
,
7WC5
,
6WH4
,
6WGT
,
7WC6
,
6WHA
,
7WC7
,
7VOD
,
7VOE
,
7WC8
,
7RAN
,
6A94
,
7WC9
,
7WC4
ZINC - Investigational
5HT2A_HUMAN
ZINC - Metabolites
5HT2A_HUMAN
HPA
ENSG00000102468-HTR2A
GeneCards
P28223
Ensembl
ENSG00000102468
,
ENST00000542664
,
ENSP00000437737
Pharos - Targets
P28223
ZINC - Predictions - Purchasable
5HT2A_HUMAN
HMDB Protein
HMDBP02658
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