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DRD1 [plasma membrane]
Stable Identifier
R-HSA-390853
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
plasma membrane
Synonyms
Dopamine receptor 1, RecName: Full=D, DRD1_HUMAN
Locations in the PathwayBrowser
Expand all
Signal Transduction (Homo sapiens)
Signaling by GPCR (Homo sapiens)
GPCR downstream signalling (Homo sapiens)
G alpha (s) signalling events (Homo sapiens)
Liganded Gs-activating GPCR acts as a GEF for Gs (Homo sapiens)
GPCR:ligand complexes that act on Gs:Heterotrimeric G-protein Gs (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
DRD1,5:DA [plasma membrane] (Homo sapiens)
DRD1,5 [plasma membrane] (Homo sapiens)
DRD1 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs:Heterotrimeric G-protein Gs (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
DRD1,5:DA [plasma membrane] (Homo sapiens)
DRD1,5 [plasma membrane] (Homo sapiens)
DRD1 [plasma membrane] (Homo sapiens)
Liganded Gs-activating GPCRs bind inactive heterotrimeric Gs (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
DRD1,5:DA [plasma membrane] (Homo sapiens)
DRD1,5 [plasma membrane] (Homo sapiens)
DRD1 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs:Heterotrimeric G-protein Gs (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
DRD1,5:DA [plasma membrane] (Homo sapiens)
DRD1,5 [plasma membrane] (Homo sapiens)
DRD1 [plasma membrane] (Homo sapiens)
The Ligand:GPCR:Gs complex dissociates (Homo sapiens)
GPCR:ligand complexes that act on Gs:Heterotrimeric G-protein Gs (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
DRD1,5:DA [plasma membrane] (Homo sapiens)
DRD1,5 [plasma membrane] (Homo sapiens)
DRD1 [plasma membrane] (Homo sapiens)
GPCRs that activate Gs [plasma membrane] (Homo sapiens)
DRD1,5 [plasma membrane] (Homo sapiens)
DRD1 [plasma membrane] (Homo sapiens)
GPCR ligand binding (Homo sapiens)
Class A/1 (Rhodopsin-like receptors) (Homo sapiens)
Amine ligand-binding receptors (Homo sapiens)
Dopamine receptors (Homo sapiens)
DRD1,5 bind DA (Homo sapiens)
DRD1,5 [plasma membrane] (Homo sapiens)
DRD1 [plasma membrane] (Homo sapiens)
DRD1,5:DA [plasma membrane] (Homo sapiens)
DRD1,5 [plasma membrane] (Homo sapiens)
DRD1 [plasma membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:P21728 DRD1
Gene Names
DRD1
Chain
chain:1-446
Reference Genes
BioGPS Gene:1812 DRD1
COSMIC (genes):DRD1 DRD1
CTD Gene:1812 DRD1
dbSNP Gene:1812 DRD1
ENSEMBL:ENSG00000184845 DRD1
HGNC:3020 DRD1
KEGG:hsa:1812 DRD1
Monarch:1812 DRD1
NCBI Gene:1812 DRD1
OMIM:126449 DRD1
UCSC:P21728 DRD1
Reference Transcript
RefSeq:NM_000794.3 DRD1
Other Identifiers
11737023_at
11737024_s_at
17002962
1812
214652_PM_at
214652_at
2888011
2888012
2888013
2888014
2888015
2888016
2888017
34550_at
8115875
A_23_P388061
GE80660
GO:0001588
GO:0001659
GO:0001661
GO:0001662
GO:0001764
GO:0001932
GO:0001963
GO:0001965
GO:0001975
GO:0003012
GO:0003013
GO:0004930
GO:0004952
GO:0005515
GO:0005634
GO:0005783
GO:0005789
GO:0005886
GO:0005929
GO:0006606
GO:0006886
GO:0006913
GO:0006936
GO:0007186
GO:0007187
GO:0007189
GO:0007190
GO:0007191
GO:0007212
GO:0007416
GO:0007612
GO:0007613
GO:0007617
GO:0007625
GO:0007626
GO:0007628
GO:0007631
GO:0008306
GO:0008542
GO:0009410
GO:0012505
GO:0014002
GO:0015872
GO:0016020
GO:0016477
GO:0019226
GO:0019228
GO:0021542
GO:0021756
GO:0021766
GO:0021853
GO:0022414
GO:0023052
GO:0030335
GO:0030425
GO:0030432
GO:0032795
GO:0034330
GO:0035106
GO:0035240
GO:0035249
GO:0042053
GO:0042220
GO:0042311
GO:0042417
GO:0042711
GO:0042734
GO:0042995
GO:0043197
GO:0043226
GO:0043268
GO:0043410
GO:0045202
GO:0045211
GO:0046323
GO:0046959
GO:0046960
GO:0048148
GO:0048856
GO:0048870
GO:0050877
GO:0051281
GO:0051584
GO:0051968
GO:0055085
GO:0060089
GO:0060134
GO:0060158
GO:0060170
GO:0060291
GO:0060292
GO:0071870
GO:0071880
GO:0097648
GO:0097730
GO:0098978
GO:0098982
GO:0099010
GO:0099171
GO:1990763
GO:2001224
HMNXSV003017464
Hs.2624.0.S2_3p_at
ILMN_1773210
M85247_at
PH_hs_0000346
TC05002083.hg
X58987_at
Participates
as a member of
DRD1,5 [plasma membrane] (Homo sapiens)
Inferred To
drd1b [plasma membrane]
(Danio rerio)
Drd1 [plasma membrane]
(Mus musculus)
Homologues of DRD1 [plasma membrane]
(Drosophila melanogaster)
DRD1 [plasma membrane]
(Bos taurus)
DRD1 [plasma membrane]
(Canis familiaris)
DRD1 [plasma membrane]
(Gallus gallus)
Octbeta1R [plasma membrane]
(Drosophila melanogaster)
Octbeta2R [plasma membrane]
(Drosophila melanogaster)
Octbeta3R [plasma membrane]
(Drosophila melanogaster)
drd1 [plasma membrane]
(Xenopus tropicalis)
Cross References
RefSeq
NP_000785.1
Guide to Pharmacology - Targets
214
OpenTargets
ENSG00000184845
ENSEMBL
ENSG00000184845
,
ENSP00000377353
,
ENST00000393752
ZINC - FDA approved
DRD1_HUMAN
ZINC - Substances
DRD1_HUMAN
ZINC - Biogenic
DRD1_HUMAN
ZINC target
P21728
PRO
P21728
GlyGen
P21728
PDB
7X2C
,
7CKZ
,
7CKX
,
7F24
,
7F1Z
,
7X2D
,
7F23
,
7F1O
,
7LJD
,
7LJC
,
7JVP
,
8IRR
,
7CKY
,
7CKW
,
7F0T
,
7JVQ
,
7CRH
,
8JXR
,
7X2F
,
7JOZ
,
7JV5
,
8JXS
ZINC - Investigational
DRD1_HUMAN
ZINC - Metabolites
DRD1_HUMAN
HPA
ENSG00000184845-DRD1
GeneCards
DRD1
Pharos - Targets
P21728
ZINC - Predictions - Purchasable
DRD1_HUMAN
HMDB Protein
HMDBP10808
Interactors (3)
Accession
#Entities
Entities
Confidence Score
Evidence (IntAct)
UniProt:Q92993 KAT5
1
KAT5 [nucleoplasm]
(R-HSA-3321979)
0.556
3
UniProt:P17252 PRKCA
8
PRKCA [cytosol]
(R-HSA-58196)
pT497,T638,S657-PRKCA [plasma membrane]
(R-HSA-4332340)
p-T497,T638,S657-PRKCA [cytosol]
(R-HSA-4332337)
PRKCA [plasma membrane]
(R-HSA-156469)
p-T497,T638,S657-PRKCA [nucleoplasm]
(R-HSA-5223292)
p-T497-PRKCA [cytosol]
(R-HSA-5218731)
PRKCA [photoreceptor disc membrane]
(R-HSA-2648987)
PRKCA [nucleoplasm]
(R-HSA-450530)
0.556
3
UniProt:Q13324-2 CRHR2
1
CRHR2-2 [plasma membrane]
(R-HSA-8937630)
0.463
2
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