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BDKRB2 [plasma membrane]
Stable Identifier
R-HSA-374255
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
plasma membrane
Synonyms
B2 bradykinin receptor, BKRB2_HUMAN
Locations in the PathwayBrowser
Expand all
Signal Transduction (Homo sapiens)
Signaling by GPCR (Homo sapiens)
GPCR downstream signalling (Homo sapiens)
G alpha (i) signalling events (Homo sapiens)
Liganded Gi-activating GPCR acts as a GEF for Gi (Homo sapiens)
Ligand:GPCR complexes that activate Gi:Heterotrimeric G-protein Gi (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
Bradykinin receptor:Bradykinin [plasma membrane] (Homo sapiens)
Bradykinin receptor [plasma membrane] (Homo sapiens)
BDKRB2 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi:Heterotrimeric G-protein Gi (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
Bradykinin receptor:Bradykinin [plasma membrane] (Homo sapiens)
Bradykinin receptor [plasma membrane] (Homo sapiens)
BDKRB2 [plasma membrane] (Homo sapiens)
Liganded Gi-activating GPCRs bind inactive heterotrimeric G-protein Gi (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
Bradykinin receptor:Bradykinin [plasma membrane] (Homo sapiens)
Bradykinin receptor [plasma membrane] (Homo sapiens)
BDKRB2 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi:Heterotrimeric G-protein Gi (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
Bradykinin receptor:Bradykinin [plasma membrane] (Homo sapiens)
Bradykinin receptor [plasma membrane] (Homo sapiens)
BDKRB2 [plasma membrane] (Homo sapiens)
The Ligand:GPCR:Gi complex dissociates (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
Bradykinin receptor:Bradykinin [plasma membrane] (Homo sapiens)
Bradykinin receptor [plasma membrane] (Homo sapiens)
BDKRB2 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi:Heterotrimeric G-protein Gi (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
Bradykinin receptor:Bradykinin [plasma membrane] (Homo sapiens)
Bradykinin receptor [plasma membrane] (Homo sapiens)
BDKRB2 [plasma membrane] (Homo sapiens)
G alpha (q) signalling events (Homo sapiens)
Liganded Gq-activating GPCRs bind inactive heterotrimeric Gq (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
Bradykinin receptor:Bradykinin [plasma membrane] (Homo sapiens)
Bradykinin receptor [plasma membrane] (Homo sapiens)
BDKRB2 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
Bradykinin receptor:Bradykinin [plasma membrane] (Homo sapiens)
Bradykinin receptor [plasma membrane] (Homo sapiens)
BDKRB2 [plasma membrane] (Homo sapiens)
Liganded Gq/11-activating GPCRs act as GEFs for Gq/11 (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
Bradykinin receptor:Bradykinin [plasma membrane] (Homo sapiens)
Bradykinin receptor [plasma membrane] (Homo sapiens)
BDKRB2 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
Bradykinin receptor:Bradykinin [plasma membrane] (Homo sapiens)
Bradykinin receptor [plasma membrane] (Homo sapiens)
BDKRB2 [plasma membrane] (Homo sapiens)
The Ligand:GPCR:Gq complex dissociates (Homo sapiens)
GPCRs that activate Gq/11 [plasma membrane] (Homo sapiens)
Bradykinin receptor [plasma membrane] (Homo sapiens)
BDKRB2 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
Bradykinin receptor:Bradykinin [plasma membrane] (Homo sapiens)
Bradykinin receptor [plasma membrane] (Homo sapiens)
BDKRB2 [plasma membrane] (Homo sapiens)
GPCR ligand binding (Homo sapiens)
Class A/1 (Rhodopsin-like receptors) (Homo sapiens)
Peptide ligand-binding receptors (Homo sapiens)
Bradykinin receptors B1 and B2 bind to bradykinin (Homo sapiens)
Bradykinin receptor [plasma membrane] (Homo sapiens)
BDKRB2 [plasma membrane] (Homo sapiens)
Bradykinin receptor:Bradykinin [plasma membrane] (Homo sapiens)
Bradykinin receptor [plasma membrane] (Homo sapiens)
BDKRB2 [plasma membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:P30411 BDKRB2
Gene Names
BDKRB2, BKR2
Chain
chain:1-391
Reference Genes
BioGPS Gene:624 BDKRB2
COSMIC (genes):BDKRB2 BDKRB2
CTD Gene:624 BDKRB2
dbSNP Gene:624 BDKRB2
ENSEMBL:ENSG00000168398 BDKRB2
HGNC:1030 BDKRB2
KEGG:hsa:624 BDKRB2
Monarch:624 BDKRB2
NCBI Gene:624 BDKRB2
OMIM:113503 BDKRB2
UCSC:P30411 BDKRB2
Reference Transcript
RefSeq:NM_000623.3 BDKRB2
Other Identifiers
11740588_at
11746532_s_at
16788023
205870_PM_at
205870_at
3550274
3550279
3550282
3550283
3550284
3550285
3550286
3550287
3550288
3550289
3550290
3550291
39309_at
39310_at
624
62824_at
7976560
A_23_P304897
GE63096
GO:0002020
GO:0003012
GO:0003013
GO:0003824
GO:0004435
GO:0004930
GO:0004947
GO:0005515
GO:0005768
GO:0005794
GO:0005886
GO:0006939
GO:0006954
GO:0007166
GO:0007169
GO:0007186
GO:0007204
GO:0008015
GO:0009651
GO:0016020
GO:0016787
GO:0019229
GO:0031410
GO:0031702
GO:0033137
GO:0042310
GO:0042311
GO:0043114
GO:0043226
GO:0043231
GO:0046982
GO:0050482
GO:0060089
GO:1902219
GO:1902239
GO:1990127
HMNXSV003035161
ILMN_1684086
PH_hs_0013287
TC14002310.hg
X86163_at
g4557358_3p_at
Participates
as a member of
Bradykinin receptor [plasma membrane] (Homo sapiens)
Inferred To
Tre1 [plasma membrane]
(Drosophila melanogaster)
moody [plasma membrane]
(Drosophila melanogaster)
Bdkrb2 [plasma membrane]
(Canis familiaris)
Bdkrb2 [plasma membrane]
(Mus musculus)
Bdkrb2 [plasma membrane]
(Rattus norvegicus)
npr-25 [plasma membrane]
(Caenorhabditis elegans)
EG:22E5.10 [plasma membrane]
(Drosophila melanogaster)
Homologues of BDKRB2 [plasma membrane]
(Drosophila melanogaster)
BDKRB2 [plasma membrane]
(Gallus gallus)
Cross References
RefSeq
NP_000614.1
Guide to Pharmacology - Targets
42
ENSEMBL
ENST00000539359
,
ENSP00000450482
,
ENSP00000438376
,
ENST00000542454
,
ENSG00000168398
,
ENST00000554311
,
ENSP00000439459
OpenTargets
ENSG00000168398
ZINC - FDA approved
BKRB2_HUMAN
ZINC - Substances
BKRB2_HUMAN
ZINC target
P30411
PRO
P30411
GlyGen
P30411
PDB
7F6H
,
7F6I
,
7F2O
ZINC - Investigational
BKRB2_HUMAN
GeneCards
BDKRB2
HPA
ENSG00000168398-BDKRB2
Pharos - Targets
P30411
ZINC - Predictions - Purchasable
BKRB2_HUMAN
HMDB Protein
HMDBP07471
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