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TAS2R8 [plasma membrane]
Stable Identifier
R-HSA-3299620
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
plasma membrane
Synonyms
Taste receptor type 2 member 8, TA2R8_HUMAN
Locations in the PathwayBrowser
Expand all
Sensory Perception (Homo sapiens)
Sensory perception of taste (Homo sapiens)
Sensory perception of sweet, bitter, and umami (glutamate) taste (Homo sapiens)
Bitter compound binds bitter taste receptor (TAS2R) (Homo sapiens)
TAS2R:GNAT3:GDP:GNB1,3:GNG13 [plasma membrane] (Homo sapiens)
TAS2R (non-orphan) [plasma membrane] (Homo sapiens)
TAS2R8 [plasma membrane] (Homo sapiens)
TAS2R:ligand:GNAT3:GDP:GNB1,3:GNG13 [plasma membrane] (Homo sapiens)
TAS2R (non-orphan):ligand [plasma membrane] (Homo sapiens)
TAS2R8:ligand [plasma membrane] (Homo sapiens)
TAS2R8 [plasma membrane] (Homo sapiens)
GNAT3 exchanges GDP for GTP in TAS2R:bitter compound:GNAT3:GDP:GNB1,3:GNG13 (Homo sapiens)
TAS2R:ligand:GNAT3:GDP:GNB1,3:GNG13 [plasma membrane] (Homo sapiens)
TAS2R (non-orphan):ligand [plasma membrane] (Homo sapiens)
TAS2R8:ligand [plasma membrane] (Homo sapiens)
TAS2R8 [plasma membrane] (Homo sapiens)
TAS2R:ligand:GNAT3:GTP:GNB1,3:GNG13 [plasma membrane] (Homo sapiens)
TAS2R (non-orphan):ligand [plasma membrane] (Homo sapiens)
TAS2R8:ligand [plasma membrane] (Homo sapiens)
TAS2R8 [plasma membrane] (Homo sapiens)
TAS2R:bitter compound:GNAT3:GTP:GNB1,3:GNG13 dissociates yielding (Homo sapiens)
TAS2R (non-orphan):ligand [plasma membrane] (Homo sapiens)
TAS2R8:ligand [plasma membrane] (Homo sapiens)
TAS2R8 [plasma membrane] (Homo sapiens)
TAS2R:ligand:GNAT3:GTP:GNB1,3:GNG13 [plasma membrane] (Homo sapiens)
TAS2R (non-orphan):ligand [plasma membrane] (Homo sapiens)
TAS2R8:ligand [plasma membrane] (Homo sapiens)
TAS2R8 [plasma membrane] (Homo sapiens)
Signal Transduction (Homo sapiens)
Signaling by GPCR (Homo sapiens)
GPCR downstream signalling (Homo sapiens)
G alpha (i) signalling events (Homo sapiens)
Liganded Gi-activating GPCR acts as a GEF for Gi (Homo sapiens)
Ligand:GPCR complexes that activate Gi:Heterotrimeric G-protein Gi (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
TAS2Rs:Bitter-tasting compounds [plasma membrane] (Homo sapiens)
TAS2Rs [plasma membrane] (Homo sapiens)
TAS2R8 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi:Heterotrimeric G-protein Gi (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
TAS2Rs:Bitter-tasting compounds [plasma membrane] (Homo sapiens)
TAS2Rs [plasma membrane] (Homo sapiens)
TAS2R8 [plasma membrane] (Homo sapiens)
Liganded Gi-activating GPCRs bind inactive heterotrimeric G-protein Gi (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
TAS2Rs:Bitter-tasting compounds [plasma membrane] (Homo sapiens)
TAS2Rs [plasma membrane] (Homo sapiens)
TAS2R8 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi:Heterotrimeric G-protein Gi (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
TAS2Rs:Bitter-tasting compounds [plasma membrane] (Homo sapiens)
TAS2Rs [plasma membrane] (Homo sapiens)
TAS2R8 [plasma membrane] (Homo sapiens)
The Ligand:GPCR:Gi complex dissociates (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
TAS2Rs:Bitter-tasting compounds [plasma membrane] (Homo sapiens)
TAS2Rs [plasma membrane] (Homo sapiens)
TAS2R8 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi:Heterotrimeric G-protein Gi (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
TAS2Rs:Bitter-tasting compounds [plasma membrane] (Homo sapiens)
TAS2Rs [plasma membrane] (Homo sapiens)
TAS2R8 [plasma membrane] (Homo sapiens)
GPCR ligand binding (Homo sapiens)
Class C/3 (Metabotropic glutamate/pheromone receptors) (Homo sapiens)
T2Rs bind bitter-tasting compounds (Homo sapiens)
TAS2Rs [plasma membrane] (Homo sapiens)
TAS2R8 [plasma membrane] (Homo sapiens)
TAS2Rs:Bitter-tasting compounds [plasma membrane] (Homo sapiens)
TAS2Rs [plasma membrane] (Homo sapiens)
TAS2R8 [plasma membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:Q9NYW2 TAS2R8
Gene Names
TAS2R8
Chain
chain:1-309
Reference Genes
BioGPS Gene:50836 TAS2R8
COSMIC (genes):TAS2R8 TAS2R8
CTD Gene:50836 TAS2R8
dbSNP Gene:50836 TAS2R8
ENSEMBL:ENSG00000121314 TAS2R8
ENSEMBL:ENSG00000121314.3 TAS2R8
ENSEMBL:ENSG00000272712.1 TAS2R8
ENSEMBL:ENSG00000277316.2 TAS2R8
HGNC:14915 TAS2R8
KEGG Gene (Homo sapiens):50836 TAS2R8
Monarch:50836 TAS2R8
NCBI Gene:50836 TAS2R8
OMIM:604794 TAS2R8
UCSC:Q9NYW2 TAS2R8
Reference Transcript
RefSeq:NM_023918.1 TAS2R8
Other Identifiers
11732972_at
16761457
221398_PM_at
221398_at
3444305
3444306
3444308
50836
7961243
ADDON002837.hg
A_23_P48022
GE499570
GO:0001580
GO:0004930
GO:0005515
GO:0005886
GO:0007165
GO:0007186
GO:0008527
GO:0016020
GO:0023052
GO:0033038
GO:0050877
GO:0050896
GO:0050909
GO:0060089
HMNXSV003013417
ILMN_1807159
ILMN_2107040
PH_hs_0014066
TC12001229.hg
TC12002760.hg
g12965173_3p_at
Participates
as a component of
TAS2R8:ligand [plasma membrane] (Homo sapiens)
as a member of
TAS2R (non-orphan) [plasma membrane] (Homo sapiens)
TAS2Rs [plasma membrane] (Homo sapiens)
Inferred To
t2r6 [plasma membrane]
(Xenopus tropicalis)
t2r37 [plasma membrane]
(Xenopus tropicalis)
t2r24 [plasma membrane]
(Xenopus tropicalis)
Homologues of TAS2R20 [plasma membrane]
(Danio rerio)
Homologues of TAS2R20 [plasma membrane]
(Gallus gallus)
Homologues of TAS2R20 [plasma membrane]
(Xenopus tropicalis)
t2r49 [plasma membrane]
(Xenopus tropicalis)
t2r52 [plasma membrane]
(Xenopus tropicalis)
rab3gap2 [plasma membrane]
(Xenopus tropicalis)
t2r45 [plasma membrane]
(Xenopus tropicalis)
t2r5 [plasma membrane]
(Xenopus tropicalis)
LOC100492238 [plasma membrane]
(Xenopus tropicalis)
LOC101747503 [plasma membrane]
(Gallus gallus)
t2r50 [plasma membrane]
(Xenopus tropicalis)
LOC100486257 [plasma membrane]
(Xenopus tropicalis)
t2r38 [plasma membrane]
(Xenopus tropicalis)
t2r10 [plasma membrane]
(Xenopus tropicalis)
t2r20 [plasma membrane]
(Xenopus tropicalis)
t2r30 [plasma membrane]
(Xenopus tropicalis)
t2r36 [plasma membrane]
(Xenopus tropicalis)
LOC101731190 [plasma membrane]
(Xenopus tropicalis)
t2r4 [plasma membrane]
(Xenopus tropicalis)
t2r17 [plasma membrane]
(Xenopus tropicalis)
t2r41 [plasma membrane]
(Xenopus tropicalis)
LOC100492564 [plasma membrane]
(Xenopus tropicalis)
tas2r4 [plasma membrane]
(Xenopus tropicalis)
t2r34 [plasma membrane]
(Xenopus tropicalis)
LOC116407540 [plasma membrane]
(Xenopus tropicalis)
t2r14 [plasma membrane]
(Xenopus tropicalis)
t2r9 [plasma membrane]
(Xenopus tropicalis)
t2r3 [plasma membrane]
(Xenopus tropicalis)
t2r19 [plasma membrane]
(Xenopus tropicalis)
TAS2R7 [plasma membrane]
(Gallus gallus)
t2r42 [plasma membrane]
(Xenopus tropicalis)
t2r35 [plasma membrane]
(Xenopus tropicalis)
t2r8 [plasma membrane]
(Xenopus tropicalis)
t2r48 [plasma membrane]
(Xenopus tropicalis)
TAS2R8 [plasma membrane]
(Bos taurus)
LOC100494566 [plasma membrane]
(Xenopus tropicalis)
t2r15 [plasma membrane]
(Xenopus tropicalis)
t2r22 [plasma membrane]
(Xenopus tropicalis)
t2r2 [plasma membrane]
(Xenopus tropicalis)
TAS2R20 [plasma membrane]
(Danio rerio)
TAS2R20 [plasma membrane]
(Xenopus tropicalis)
tas2r39 [plasma membrane]
(Xenopus tropicalis)
LOC108648843 [plasma membrane]
(Xenopus tropicalis)
t2r53 [plasma membrane]
(Xenopus tropicalis)
t2r43 [plasma membrane]
(Xenopus tropicalis)
t2r13 [plasma membrane]
(Xenopus tropicalis)
TAS2R1a [plasma membrane]
(Danio rerio)
tas2r7 [plasma membrane]
(Xenopus tropicalis)
TAS2R40 [plasma membrane]
(Gallus gallus)
t2r54 [plasma membrane]
(Xenopus tropicalis)
Cross References
RefSeq
NP_076407.1
Guide to Pharmacology - Targets
664
OpenTargets
ENSG00000121314
HPA
ENSG00000121314-TAS2R8
GeneCards
Q9NYW2
Ensembl
ENSP00000484163
,
ENSG00000121314
,
ENSG00000277316
,
ENSP00000461158
,
ENST00000572823
,
ENST00000240615
,
ENST00000610444
,
ENSP00000240615
,
ENSG00000272712
PRO
Q9NYW2
Pharos - Targets
Q9NYW2
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