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ABCB1 [plasma membrane]
Stable Identifier
R-HSA-1457534
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
plasma membrane
Synonyms
MDR1, Multidrug resistance protein 1, MDR1_HUMAN, P-glycoprotein, PgP
Locations in the PathwayBrowser
Expand all
Drug ADME (Homo sapiens)
Abacavir ADME (Homo sapiens)
Abacavir transmembrane transport (Homo sapiens)
abacavir [cytosol] + ATP + H2O => abacavir[extracellular] + ADP + phosphate (Homo sapiens)
ABCB1 [plasma membrane] (Homo sapiens)
Atorvastatin ADME (Homo sapiens)
ABCB1,ABCC2 transport ATVs from cytosol to extracellular region (Homo sapiens)
ABCB1,ABCC2 [plasma membrane] (Homo sapiens)
ABCB1 [plasma membrane] (Homo sapiens)
Prednisone ADME (Homo sapiens)
ABCB1 transports PREDN,PREDL out of hepatic cells (Homo sapiens)
ABCB1 [plasma membrane] (Homo sapiens)
ABCB1 transports PREDN,PREDL out of kidney cells (Homo sapiens)
ABCB1 [plasma membrane] (Homo sapiens)
ABCB1 transports xenobiotics out of the cell (Homo sapiens)
ABCB1 [plasma membrane] (Homo sapiens)
ABCB1:ABCB1 inhibitors [plasma membrane] (Homo sapiens)
ABCB1 [plasma membrane] (Homo sapiens)
Transport of small molecules (Homo sapiens)
ABC-family proteins mediated transport (Homo sapiens)
ABCA8,B1,B5 transport xenobiotics from cytosol to extracellular region (Homo sapiens)
ABCA8/B1/B5 [plasma membrane] (Homo sapiens)
ABCB1 [plasma membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:P08183 ABCB1
Gene Names
ABCB1, MDR1, PGY1
Chain
chain:1-1280
Reference Genes
BioGPS Gene:5243 ABCB1
COSMIC (genes):ABCB1 ABCB1
CTD Gene:5243 ABCB1
dbSNP Gene:5243 ABCB1
ENSEMBL:ENSG00000085563 ABCB1
HGNC:40 ABCB1
KEGG:hsa:5243 ABCB1
Monarch:5243 ABCB1
NCBI Gene:5243 ABCB1
OMIM:171050 ABCB1
UCSC:P08183 ABCB1
Reference Transcript
RefSeq:NM_000927.4 ABCB1
Other Identifiers
11730907_a_at
11759046_at
11759047_x_at
11759048_at
1575_at
1576_g_at
1682_s_at
17059491
209993_PM_at
209993_at
209994_PM_s_at
209994_s_at
243951_PM_at
243951_at
3060121
3060140
3060184
3060185
3060186
3060187
3060188
3060189
3060190
3060191
3060194
3060195
3060196
3060198
3060199
3060200
3060201
3060203
3060204
3060205
3060207
3060208
3060210
3060211
3060212
3060213
3060214
3060215
3060216
3060217
3060218
3060221
3060223
3060224
3060226
3060227
3060228
3060230
3060231
3060232
3060233
3060234
3060235
3060236
3060242
5243
60295_at
8140782
A_23_P82523
A_33_P3332414
GE57835
GO:0000086
GO:0003013
GO:0003824
GO:0005215
GO:0005515
GO:0005524
GO:0005737
GO:0005886
GO:0006805
GO:0006869
GO:0008559
GO:0009410
GO:0009986
GO:0015562
GO:0016020
GO:0016324
GO:0016787
GO:0016887
GO:0022857
GO:0031625
GO:0042626
GO:0042910
GO:0043226
GO:0045332
GO:0046865
GO:0046943
GO:0055085
GO:0061024
GO:0070062
GO:0070633
GO:0072089
GO:0090554
GO:0090555
GO:0098591
GO:0099038
GO:0099040
GO:0140115
GO:0140326
GO:0140328
GO:0140359
GO:0140657
GO:0150104
GO:1905039
GO:1990961
GO:1990962
GO:2001225
HMNXSV003054433
Hs.129467.0.A1_3p_at
ILMN_1812070
ILMN_2094875
M14758_at
PH_hs_0001839
TC07001579.hg
TC07003053.hg
X58723_at
g2353263_3p_at
g9961253_3p_s_at
p33892
Participates
as a member of
ABCB1,ABCC2 [plasma membrane] (Homo sapiens)
ABCA8/B1/B5 [plasma membrane] (Homo sapiens)
as a component of
ABCB1:ABCB1 inhibitors [plasma membrane] (Homo sapiens)
Inferred To
Homologues of ABCB1 [plasma membrane]
(Dictyostelium discoideum)
Homologues of ABCB1 [plasma membrane]
(Schizosaccharomyces pombe)
ABCB1 [plasma membrane]
(Bos taurus)
ABCB1 [plasma membrane]
(Canis familiaris)
ABCB1 [plasma membrane]
(Dictyostelium discoideum)
ABCB1 [plasma membrane]
(Gallus gallus)
ABCB1 [plasma membrane]
(Mus musculus)
ABCB1 [plasma membrane]
(Plasmodium falciparum)
ABCB1 [plasma membrane]
(Rattus norvegicus)
ABCB1 [plasma membrane]
(Schizosaccharomyces pombe)
LOC100522267 [plasma membrane]
(Sus scrofa)
Cross References
ZINC - World Drugs
MDR1_HUMAN
Guide to Pharmacology - Targets
768
OpenTargets
ENSG00000085563
ENSEMBL
ENSP00000478255
,
ENSP00000444095
,
ENST00000265724
,
ENST00000543898
,
ENST00000622132
,
ENSP00000265724
ZINC - FDA approved
MDR1_HUMAN
ZINC - Substances
MDR1_HUMAN
ZINC - Biogenic
MDR1_HUMAN
ZINC target
P08183
PRO
P08183
GlyGen
P08183
PDB
7O9W
,
8Y6I
,
6FN4
,
7A6C
,
7A69
,
6QEX
,
8Y6H
,
7A65
,
6C0V
,
6FN1
,
7A6E
,
7A6F
ZINC - Investigational
MDR1_HUMAN
ZINC - Metabolites
MDR1_HUMAN
IntEnz
7.6.2.1
HPA
ENSG00000085563-ABCB1
Pharos - Targets
P08183
ZINC - Predictions - Purchasable
MDR1_HUMAN
Orphanet
ABCB1
HMDB Protein
HMDBP02101
Interactors (2)
Accession
#Entities
Entities
Confidence Score
Evidence (IntAct)
UniProt:P17931 LGALS3
3
LGALS3 [ficolin-1-rich granule membrane]
(R-HSA-6803307)
LGALS3 [plasma membrane]
(R-HSA-879445)
LGALS3 [secretory granule membrane]
(R-HSA-6803327)
0.527
3
UniProt:Q99496 RNF2
1
RNF2 [nucleoplasm]
(R-HSA-389119)
0.508
2
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