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avapritinib [cytosol]
Stable Identifier
R-ALL-9671491
Type
ChemicalDrug
Compartment
cytosol
Synonyms
BLU285, BLU-285
Locations in the PathwayBrowser
for Species:
Homo sapiens
Bos taurus
Caenorhabditis elegans
Canis familiaris
Danio rerio
Drosophila melanogaster
Gallus gallus
Mus musculus
Rattus norvegicus
Sus scrofa
Xenopus tropicalis
Expand all
Signal Transduction (Bos taurus)
Signaling by Receptor Tyrosine Kinases (Bos taurus)
Signaling by PDGF (Bos taurus)
Autophosphorylation of PDGF alpha receptors (Bos taurus)
PDGFR:type I PDGFR-binding TKIs [plasma membrane] (Bos taurus)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
PDGFRs bind type I TKI (Bos taurus)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
PDGFR:type I PDGFR-binding TKIs [plasma membrane] (Bos taurus)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
Signaling by SCF-KIT (Bos taurus)
Autophosphorylation of KIT (Bos taurus)
KIT:sSCF dimer:KIT:type I KIT binding TKIs: [plasma membrane] (Bos taurus)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
KIT binds type I TKIs (Bos taurus)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
KIT:sSCF dimer:KIT:type I KIT binding TKIs: [plasma membrane] (Bos taurus)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
Signal Transduction (Caenorhabditis elegans)
Signaling by Receptor Tyrosine Kinases (Caenorhabditis elegans)
Signaling by PDGF (Caenorhabditis elegans)
Autophosphorylation of PDGF alpha receptors (Caenorhabditis elegans)
PDGFR:type I PDGFR-binding TKIs [plasma membrane] (Caenorhabditis elegans)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
PDGFRs bind type I TKI (Caenorhabditis elegans)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
PDGFR:type I PDGFR-binding TKIs [plasma membrane] (Caenorhabditis elegans)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
Signal Transduction (Canis familiaris)
Signaling by Receptor Tyrosine Kinases (Canis familiaris)
Signaling by PDGF (Canis familiaris)
Autophosphorylation of PDGF alpha receptors (Canis familiaris)
PDGFR:type I PDGFR-binding TKIs [plasma membrane] (Canis familiaris)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
PDGFRs bind type I TKI (Canis familiaris)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
PDGFR:type I PDGFR-binding TKIs [plasma membrane] (Canis familiaris)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
Signaling by SCF-KIT (Canis familiaris)
Autophosphorylation of KIT (Canis familiaris)
KIT:sSCF dimer:KIT:type I KIT binding TKIs: [plasma membrane] (Canis familiaris)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
KIT binds type I TKIs (Canis familiaris)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
KIT:sSCF dimer:KIT:type I KIT binding TKIs: [plasma membrane] (Canis familiaris)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
Signal Transduction (Danio rerio)
Signaling by Receptor Tyrosine Kinases (Danio rerio)
Signaling by PDGF (Danio rerio)
Autophosphorylation of PDGF alpha receptors (Danio rerio)
PDGFR:type I PDGFR-binding TKIs [plasma membrane] (Danio rerio)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
PDGFRs bind type I TKI (Danio rerio)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
PDGFR:type I PDGFR-binding TKIs [plasma membrane] (Danio rerio)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
Signaling by SCF-KIT (Danio rerio)
Autophosphorylation of KIT (Danio rerio)
KIT:sSCF dimer:KIT:type I KIT binding TKIs: [plasma membrane] (Danio rerio)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
KIT binds type I TKIs (Danio rerio)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
KIT:sSCF dimer:KIT:type I KIT binding TKIs: [plasma membrane] (Danio rerio)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
Signal Transduction (Drosophila melanogaster)
Signaling by Receptor Tyrosine Kinases (Drosophila melanogaster)
Signaling by PDGF (Drosophila melanogaster)
Autophosphorylation of PDGF alpha receptors (Drosophila melanogaster)
PDGFR:type I PDGFR-binding TKIs [plasma membrane] (Drosophila melanogaster)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
PDGFRs bind type I TKI (Drosophila melanogaster)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
PDGFR:type I PDGFR-binding TKIs [plasma membrane] (Drosophila melanogaster)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
Signal Transduction (Gallus gallus)
Signaling by Receptor Tyrosine Kinases (Gallus gallus)
Signaling by PDGF (Gallus gallus)
Autophosphorylation of PDGF alpha receptors (Gallus gallus)
PDGFR:type I PDGFR-binding TKIs [plasma membrane] (Gallus gallus)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
PDGFRs bind type I TKI (Gallus gallus)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
PDGFR:type I PDGFR-binding TKIs [plasma membrane] (Gallus gallus)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
Signaling by SCF-KIT (Gallus gallus)
Autophosphorylation of KIT (Gallus gallus)
KIT:sSCF dimer:KIT:type I KIT binding TKIs: [plasma membrane] (Gallus gallus)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
KIT binds type I TKIs (Gallus gallus)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
KIT:sSCF dimer:KIT:type I KIT binding TKIs: [plasma membrane] (Gallus gallus)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
Disease (Homo sapiens)
Diseases of signal transduction by growth factor receptors and second messengers (Homo sapiens)
Signaling by KIT in disease (Homo sapiens)
KIT mutants bind TKIs (Homo sapiens)
KIT mutants bind type I TKIs (Homo sapiens)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
type I sensitive KIT mutants:type I TKIs [plasma membrane] (Homo sapiens)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
Signaling by PDGFR in disease (Homo sapiens)
PDGFR mutants bind TKIs (Homo sapiens)
PDGFR mutants bind type I TKIs (Homo sapiens)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
type I sensitive PDGFR mutants:type I TKIs [plasma membrane] (Homo sapiens)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
Signal Transduction (Homo sapiens)
Signaling by Receptor Tyrosine Kinases (Homo sapiens)
Signaling by PDGF (Homo sapiens)
Autophosphorylation of PDGF alpha receptors (Homo sapiens)
PDGFR:type I PDGFR-binding TKIs [plasma membrane] (Homo sapiens)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
PDGFRs bind type I TKI (Homo sapiens)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
PDGFR:type I PDGFR-binding TKIs [plasma membrane] (Homo sapiens)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
Signaling by SCF-KIT (Homo sapiens)
Autophosphorylation of KIT (Homo sapiens)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
KIT:sSCF dimer:KIT:type I KIT binding TKIs: [plasma membrane] (Homo sapiens)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
KIT binds type I TKIs (Homo sapiens)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
KIT:sSCF dimer:KIT:type I KIT binding TKIs: [plasma membrane] (Homo sapiens)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
Signal Transduction (Mus musculus)
Signaling by Receptor Tyrosine Kinases (Mus musculus)
Signaling by PDGF (Mus musculus)
Autophosphorylation of PDGF alpha receptors (Mus musculus)
PDGFR:type I PDGFR-binding TKIs [plasma membrane] (Mus musculus)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
PDGFRs bind type I TKI (Mus musculus)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
PDGFR:type I PDGFR-binding TKIs [plasma membrane] (Mus musculus)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
Signaling by SCF-KIT (Mus musculus)
Autophosphorylation of KIT (Mus musculus)
KIT:sSCF dimer:KIT:type I KIT binding TKIs: [plasma membrane] (Mus musculus)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
KIT binds type I TKIs (Mus musculus)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
KIT:sSCF dimer:KIT:type I KIT binding TKIs: [plasma membrane] (Mus musculus)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
Signal Transduction (Rattus norvegicus)
Signaling by Receptor Tyrosine Kinases (Rattus norvegicus)
Signaling by PDGF (Rattus norvegicus)
Autophosphorylation of PDGF alpha receptors (Rattus norvegicus)
PDGFR:type I PDGFR-binding TKIs [plasma membrane] (Rattus norvegicus)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
PDGFRs bind type I TKI (Rattus norvegicus)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
PDGFR:type I PDGFR-binding TKIs [plasma membrane] (Rattus norvegicus)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
Signaling by SCF-KIT (Rattus norvegicus)
Autophosphorylation of KIT (Rattus norvegicus)
KIT:sSCF dimer:KIT:type I KIT binding TKIs: [plasma membrane] (Rattus norvegicus)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
KIT binds type I TKIs (Rattus norvegicus)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
KIT:sSCF dimer:KIT:type I KIT binding TKIs: [plasma membrane] (Rattus norvegicus)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
Signal Transduction (Sus scrofa)
Signaling by Receptor Tyrosine Kinases (Sus scrofa)
Signaling by PDGF (Sus scrofa)
Autophosphorylation of PDGF alpha receptors (Sus scrofa)
PDGFR:type I PDGFR-binding TKIs [plasma membrane] (Sus scrofa)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
PDGFRs bind type I TKI (Sus scrofa)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
PDGFR:type I PDGFR-binding TKIs [plasma membrane] (Sus scrofa)
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
avapritinib [cytosol]
Signaling by SCF-KIT (Sus scrofa)
Autophosphorylation of KIT (Sus scrofa)
KIT:sSCF dimer:KIT:type I KIT binding TKIs: [plasma membrane] (Sus scrofa)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
KIT binds type I TKIs (Sus scrofa)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
KIT:sSCF dimer:KIT:type I KIT binding TKIs: [plasma membrane] (Sus scrofa)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
Signal Transduction (Xenopus tropicalis)
Signaling by Receptor Tyrosine Kinases (Xenopus tropicalis)
Signaling by SCF-KIT (Xenopus tropicalis)
Autophosphorylation of KIT (Xenopus tropicalis)
KIT:sSCF dimer:KIT:type I KIT binding TKIs: [plasma membrane] (Xenopus tropicalis)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
KIT binds type I TKIs (Xenopus tropicalis)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
KIT:sSCF dimer:KIT:type I KIT binding TKIs: [plasma membrane] (Xenopus tropicalis)
type I KIT binding TKIs [cytosol]
avapritinib [cytosol]
External Reference Information
External Reference
avapritinib [Guide to Pharmacology:10368]
Participates
as a member of
type I KIT binding TKIs [cytosol]
type I PDGFR-binding tyrosine kinase inhibitors [cytosol]
Disease
Name
Identifier
Synonyms
cancer
DOID:162
malignant tumor, malignant neoplasm, primary cancer
Cross References
PharmacoDB
PDBC31443
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