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dabrafenib mesylate [cytosol]
Stable Identifier
R-ALL-6802252
Type
ChemicalDrug
Compartment
cytosol
Locations in the PathwayBrowser
Expand all
Disease (Homo sapiens)
Diseases of signal transduction by growth factor receptors and second messengers (Homo sapiens)
Oncogenic MAPK signaling (Homo sapiens)
Signaling by high-kinase activity BRAF mutants (Homo sapiens)
Inhibitors bind and inhibit highly active BRAF mutants (Homo sapiens)
BRAF inhibitors [cytosol]
dabrafenib mesylate [cytosol]
BRAF inhibitors:high kinase activity BRAF mutants [cytosol] (Homo sapiens)
BRAF inhibitors [cytosol]
dabrafenib mesylate [cytosol]
Literature References
PubMed ID
Title
Journal
Year
23881668
Dabrafenib: first global approval
Garnock-Jones, KP
,
Ballantyne, AD
Drugs
2013
External Reference Information
External Reference
dabrafenib [Guide to Pharmacology:6494]
Participates
as a member of
BRAF inhibitors [cytosol]
Disease
Name
Identifier
Synonyms
melanoma
DOID:1909
Naevocarcinoma, melanoma, melanoma, malignant melanoma, morphology (morphologic abnormality), malignant melanoma NOS (morphologic abnormality), malignant melanoma (disorder), malignant melanoma, malignant melanoma, malignant melanoma, malignant melanoma
cancer
DOID:162
malignant tumor, malignant neoplasm, primary cancer
Cross References
ChEBI
75048
,
75045
Pharos - Ligands
FNCP32ZHDMMP
PharmacoDB
PDBC02065
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