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CNR2 [plasma membrane]
Stable Identifier
R-HSA-419372
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
plasma membrane
Synonyms
Cannabinoid receptor 2, CNR2_HUMAN
Locations in the PathwayBrowser
Expand all
Signal Transduction (Homo sapiens)
Signaling by GPCR (Homo sapiens)
GPCR downstream signalling (Homo sapiens)
G alpha (i) signalling events (Homo sapiens)
Liganded Gi-activating GPCR acts as a GEF for Gi (Homo sapiens)
Ligand:GPCR complexes that activate Gi:Heterotrimeric G-protein Gi (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
CNRs:Cannabinoids [plasma membrane] (Homo sapiens)
CNRs [plasma membrane] (Homo sapiens)
CNR2 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi:Heterotrimeric G-protein Gi (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
CNRs:Cannabinoids [plasma membrane] (Homo sapiens)
CNRs [plasma membrane] (Homo sapiens)
CNR2 [plasma membrane] (Homo sapiens)
Liganded Gi-activating GPCRs bind inactive heterotrimeric G-protein Gi (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
CNRs:Cannabinoids [plasma membrane] (Homo sapiens)
CNRs [plasma membrane] (Homo sapiens)
CNR2 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi:Heterotrimeric G-protein Gi (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
CNRs:Cannabinoids [plasma membrane] (Homo sapiens)
CNRs [plasma membrane] (Homo sapiens)
CNR2 [plasma membrane] (Homo sapiens)
The Ligand:GPCR:Gi complex dissociates (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
CNRs:Cannabinoids [plasma membrane] (Homo sapiens)
CNRs [plasma membrane] (Homo sapiens)
CNR2 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi:Heterotrimeric G-protein Gi (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gi [plasma membrane] (Homo sapiens)
CNRs:Cannabinoids [plasma membrane] (Homo sapiens)
CNRs [plasma membrane] (Homo sapiens)
CNR2 [plasma membrane] (Homo sapiens)
GPCR ligand binding (Homo sapiens)
Class A/1 (Rhodopsin-like receptors) (Homo sapiens)
CNRs bind CNR agonists (Homo sapiens)
CNRs [plasma membrane] (Homo sapiens)
CNR2 [plasma membrane] (Homo sapiens)
CNRs:CNR agonists [plasma membrane] (Homo sapiens)
CNRs [plasma membrane] (Homo sapiens)
CNR2 [plasma membrane] (Homo sapiens)
Cannabinoid receptors can bind cannabinoids (Homo sapiens)
CNRs [plasma membrane] (Homo sapiens)
CNR2 [plasma membrane] (Homo sapiens)
CNRs:Cannabinoids [plasma membrane] (Homo sapiens)
CNRs [plasma membrane] (Homo sapiens)
CNR2 [plasma membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:P34972 CNR2
Gene Names
CNR2, CB2A, CB2B
Chain
chain:1-360
Reference Genes
BioGPS Gene:1269 CNR2
COSMIC (genes):CNR2 CNR2
CTD Gene:1269 CNR2
dbSNP Gene:1269 CNR2
ENSEMBL:ENSG00000188822 CNR2
ENSEMBL_homo_sapiens_GENE:ENSG00000188822.8 CNR2
HGNC:2160 CNR2
KEGG Gene (Homo sapiens):1269 CNR2
Monarch:1269 CNR2
NCBI Gene:1269 CNR2
OMIM:605051 CNR2
UCSC:P34972 CNR2
Reference Transcript
RefSeq:XM_017000261.1 CNR2
RefSeq:NM_001841.2 CNR2
RefSeq:XM_011540629.2 CNR2
Other Identifiers
11740101_at
1269
16683460
206586_PM_at
206586_at
2401657
2401658
2401659
2401660
2401661
2401662
2401663
2401664
36771_at
4044361
4044364
4044365
4044366
4044367
4044368
4044369
4044370
4044371
4044379
4044388
42034_at
71015_r_at
78943_at
7913705
A_23_P310931
A_32_P48054
GE508359
GE80052
GE907178
GO:0001975
GO:0002376
GO:0004930
GO:0004949
GO:0005515
GO:0005737
GO:0005783
GO:0005886
GO:0006954
GO:0006955
GO:0007165
GO:0007186
GO:0007187
GO:0007189
GO:0016020
GO:0019222
GO:0023052
GO:0030425
GO:0030595
GO:0031234
GO:0032229
GO:0032496
GO:0033004
GO:0038171
GO:0042995
GO:0043025
GO:0043204
GO:0043226
GO:0045759
GO:0048870
GO:0060089
HMNXSV003026643
HMNXSV003040873
PH_hs_0004925
TC01002353.hg
X74328_rna1_at
g4502928_3p_at
Participates
as a member of
CNRs [plasma membrane] (Homo sapiens)
Inferred To
Cnr2 [plasma membrane]
(Mus musculus)
Cnr2 [plasma membrane]
(Rattus norvegicus)
CNR2 [plasma membrane]
(Bos taurus)
CNR2 [plasma membrane]
(Canis familiaris)
CNR2 [plasma membrane]
(Gallus gallus)
CNR2 [plasma membrane]
(Sus scrofa)
cnr2 [plasma membrane]
(Xenopus tropicalis)
cb2b [plasma membrane]
(Danio rerio)
Cross References
RefSeq
XP_011538931.1
,
NP_001832.1
,
XP_016855750.1
ZINC - World Drugs
CNR2_HUMAN
Guide to Pharmacology - Targets
57
OpenTargets
ENSG00000188822
ZINC - FDA approved
CNR2_HUMAN
ZINC - Substances
CNR2_HUMAN
ZINC - Biogenic
CNR2_HUMAN
ZINC target
P34972
PRO
P34972
PDB
6KPC
,
8GUT
,
8GUR
,
5ZTY
,
8GUS
,
6KPF
,
8GUQ
,
6PT0
,
2KI9
ZINC - Investigational
CNR2_HUMAN
ZINC - Metabolites
CNR2_HUMAN
HPA
ENSG00000188822-CNR2
GeneCards
P34972
Ensembl
ENSG00000188822
,
ENSP00000363596
,
ENST00000374472
Pharos - Targets
P34972
Orphanet
28455
ZINC - Predictions - Purchasable
CNR2_HUMAN
Interactors (4)
Accession
#Entities
Entities
Confidence Score
Evidence (IntAct)
UniProt:Q96AA3 RFT1
2
RFT1 R67C [endoplasmic reticulum membrane]
(R-HSA-4570578)
RFT1 [endoplasmic reticulum membrane]
(R-HSA-449255)
0.556
3
UniProt:Q13501 SQSTM1
7
SQSTM1(2-251)-p-7Y-ALK(1058-1620) fusion [cytosol]
(R-HSA-9711967)
SQSTM1(2-251)-ALK(1058-1620) fusion [cytosol]
(R-HSA-9711954)
K7 ub-SQSTM1 [cytosol]
(R-HSA-9759088)
p-S349 SQSTM1 [cytosol]
(R-HSA-9766524)
ub K420 p-S349 SQSTM1 [cytosol]
(R-HSA-9766536)
SQSTM1 [nucleoplasm]
(R-HSA-210961)
SQSTM1 [cytosol]
(R-HSA-193937)
0.556
5
UniProt:Q15848 ADIPOQ
1
ADIPOQ [extracellular region]
(R-HSA-1183052)
0.556
3
UniProt:P21964 COMT
2
COMT [plasma membrane]
(R-HSA-379386)
COMT [cytosol]
(R-HSA-175974)
0.556
3
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